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2006

Journal Article

beta-Secretase inhibitors: Modification at the P-4 position and improvement of inhibitory activity in cultured cells

Hamada, Yoshio, Igawa, Naoto, Ikari, Hayato, Ziora, Zyta, Nguyen, Jeffrey-Tri, Yamani, Abdellah, Hidaka, Koushi, Kimura, Tooru, Saito, Kazuki, Hayashi, Yoshio, Ebina, Maiko, Ishiura, Shoichi and Kiso, Yoshiaki (2006). beta-Secretase inhibitors: Modification at the P-4 position and improvement of inhibitory activity in cultured cells. Bioorganic and Medicinal Chemistry Letters, 16 (16), 4354-4359. doi: 10.1016/j.bmcl.2006.05.046

beta-Secretase inhibitors: Modification at the P-4 position and improvement of inhibitory activity in cultured cells

2006

Journal Article

Small-sized BACE1 inhibitors

Zyta, Ziora, Tooru, KImura and Yoshiaki, Kiso (2006). Small-sized BACE1 inhibitors. Drugs of the Future, 31 (1), 53-63. doi: 10.1358/dof.2006.031.01.957326

Small-sized BACE1 inhibitors

2006

Journal Article

Phenylthionorstatine as a transition-state mimic in BACE1 inhibitors

Ziora Zyta, Kasai Soko, Hidaka Koushi, Nagamine Ayaka, Kimura Tooru, Saito K., Hayashi Yoshio and Kiso Yoshiaki (2006). Phenylthionorstatine as a transition-state mimic in BACE1 inhibitors. Peptide Science, 2006, 237-238.

Phenylthionorstatine as a transition-state mimic in BACE1 inhibitors

2001

Journal Article

Synthesis and spectroscopic characterization of protected N-phosphonomethylglycine dipeptides

Ziora, Zyta, Kafarski, Pawel, Holband, Jolanta and Wojcik, Grazyna (2001). Synthesis and spectroscopic characterization of protected N-phosphonomethylglycine dipeptides. Journal of Peptide Science, 7 (9), 466-473. doi: 10.1002/psc.340

Synthesis and spectroscopic characterization of protected N-phosphonomethylglycine dipeptides

2001

Journal Article

Conformational polymorphism of diethyl 1-(phthalylglycyloxy)-2-phthalylaminoethenephosphonate

Holband, J, Wojcik, G, Ziora, Z and Kafarski, P (2001). Conformational polymorphism of diethyl 1-(phthalylglycyloxy)-2-phthalylaminoethenephosphonate. Journal of Molecular Structure, 595 (1-3), 167-174. doi: 10.1016/S0022-2860(01)00521-X

Conformational polymorphism of diethyl 1-(phthalylglycyloxy)-2-phthalylaminoethenephosphonate

2000

Journal Article

H-1 NMR studies of rotational isomerism in phosphonic analogues of aspartic acid

Jedrzejczyk, D, Ziora, Z and Kafarski, P (2000). H-1 NMR studies of rotational isomerism in phosphonic analogues of aspartic acid. Magnetic Resonance in Chemistry, 38 (5), 370-374. doi: 10.1002/1097-458x(200005)38:53.0.co;2-m

H-1 NMR studies of rotational isomerism in phosphonic analogues of aspartic acid

2000

Journal Article

Reactions of N-phthalylamino acid chlorides with trialkyl phosphites

Ziora, Zyta, Maly, Alina, Lejczak, Barbara, Kafarski, Pawel, Holband, Jolanta and Wójcik, Grażyna (2000). Reactions of N-phthalylamino acid chlorides with trialkyl phosphites. Heteroatom Chemistry, 11 (3), 232-239. doi: 10.1002/(sici)1098-1071(2000)11:33.0.co;2-u

Reactions of N-phthalylamino acid chlorides with trialkyl phosphites

1999

Journal Article

Synthesis of triethyl N-formyl-N-phosphonomethylglycinate and diethyl N-formyl-N- phosphonomethylglycine and studies of their rotational conformers by dynamic NMR

Ziora, Z, Cierpicki, T, Grembecka, J and Kafarski, P (1999). Synthesis of triethyl N-formyl-N-phosphonomethylglycinate and diethyl N-formyl-N- phosphonomethylglycine and studies of their rotational conformers by dynamic NMR. Journal of Chemical Research (2), 68-69A. doi: 10.1039/a806474a

Synthesis of triethyl N-formyl-N-phosphonomethylglycinate and diethyl N-formyl-N- phosphonomethylglycine and studies of their rotational conformers by dynamic NMR

1999

Journal Article

Reaction of N-Phtalylamino Acid Chlorides with Trialkyl Phosphites

Ziora, Zyta, Maly, Alina, Lejczak, Barbara and Kafarski, Paweł (1999). Reaction of N-Phtalylamino Acid Chlorides with Trialkyl Phosphites. Phosphorus, Sulfur, and Silicon and the Related Elements, 147 (1), 145-145. doi: 10.1080/10426509908053553

Reaction of N-Phtalylamino Acid Chlorides with Trialkyl Phosphites