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2002 Journal Article Recent discovery and development of protein tyrosine phosphatase inhibitorsBlaskovich, Mark A. and Kim, Hwa-Ok (2002). Recent discovery and development of protein tyrosine phosphatase inhibitors. Expert Opinion on Therapeutic Patents, 12 (6), 871-905. doi: 10.1517/13543776.12.6.871 |
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2002 Journal Article Preparation of 1-[N-Benzyloxycarbonyl-(1S)-1-amino-2-oxoethyl]-4-methyl-2,6,7-trioxabicyclo-[2.2.2]octaneRose, Nicholas G.W., Blaskovich, Mark A., Evindar, Ghotas, Wilkinson, Scott, Luo, Yue, Reid, C. and Lajoie, Gilles A. (2002). Preparation of 1-[N-Benzyloxycarbonyl-(1S)-1-amino-2-oxoethyl]-4-methyl-2,6,7-trioxabicyclo-[2.2.2]octane. Organic syntheses, 79, 216-221. doi: 10.1002/0471264180.os079.26 |
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2002 Journal Article Preparation of 1-[N-benzyloxycarbonyl-(1S)-1-amino-2-oxoethyl]-4-methyl-2,6,7-trioxabicyclo[2.2.2] octane: [Carbamic acid, [1-(4-methyl-2,6,7-trioxabicyclo[2.2.2]oct-1-yl)-2-oxoethyl]-, phenylmethyl ester, (S)-]Rose, Nicholas G. W., Blaskovich, Mark A., Evindar, Ghotas, Wilkinson, Scott, Luo, Yue, Fishlock, Dan, Reid, Chris, Lajoie, Gilles A., Gordon, Richard S. and Holmes, Andrew B. (2002). Preparation of 1-[N-benzyloxycarbonyl-(1S)-1-amino-2-oxoethyl]-4-methyl-2,6,7-trioxabicyclo[2.2.2] octane: [Carbamic acid, [1-(4-methyl-2,6,7-trioxabicyclo[2.2.2]oct-1-yl)-2-oxoethyl]-, phenylmethyl ester, (S)-]. Organic Syntheses, 79 doi: 10.15227/orgsyn.079.0216 |
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2001 Journal Article Synthesis of enantiomerically enriched beta,gamma-unsaturated-alpha-amino acidsRose, Ngw, Blaskovich, MA, Wong, A and Lajoie, GA (2001). Synthesis of enantiomerically enriched beta,gamma-unsaturated-alpha-amino acids. Tetrahedron, 57 (8), 1497-1507. doi: 10.1016/S0040-4020(00)01146-7 |
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1999 Journal Article Stereoselective synthesis of beta-substituted alpha,beta-diamino acids from beta-hydroxy amino acidsLuo, Y, Blaskovich, MA and Lajoie, GA (1999). Stereoselective synthesis of beta-substituted alpha,beta-diamino acids from beta-hydroxy amino acids. Journal of Organic Chemistry, 64 (16), 6106-6111. doi: 10.1021/jo9904718 |
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1998 Journal Article Highly efficient and versatile synthesis of libraries of constrained beta-strand mimeticsOgbu, CO, Qabar, MN, Boatman, PD, Urban, J, Meara, JP, Ferguson, MD, Tulinsky, J, Lum, C, Babu, S, Blaskovich, MA, Nakanishi, H, Ruan, FQ, Cao, BL, Minarik, R, Little, T, Nelson, S, Nguyen, M, Gall, A and Kahn, M (1998). Highly efficient and versatile synthesis of libraries of constrained beta-strand mimetics. Bioorganic & Medicinal Chemistry Letters, 8 (17), 2321-2326. doi: 10.1016/S0960-894X(98)00420-X |
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1998 Journal Article Polymer-supported acetylide addition to hexa-2,4-dienalBlaskovich, MA and Kahn, M (1998). Polymer-supported acetylide addition to hexa-2,4-dienal. Synthesis-Stuttgart (7), 965-966. |
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1998 Journal Article Stereoselective synthesis of Threo and Erythro beta-hydroxy and beta-disubstituted-beta-hydroxy alpha-amino acids (vol 63, pg 3635, 1998)Blaskovich, MA, Evindar, G, Rose, NGW, Wilkinson, S, Luo, Y and Lajoie, GA (1998). Stereoselective synthesis of Threo and Erythro beta-hydroxy and beta-disubstituted-beta-hydroxy alpha-amino acids (vol 63, pg 3635, 1998). Journal of Organic Chemistry, 63 (13), 4560-4560. doi: 10.1021/jo9849853 |
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1998 Journal Article Regiocontrol in alkylations of alpha-silyl hydrazonesBlaskovich, MA and Rickards, RW (1998). Regiocontrol in alkylations of alpha-silyl hydrazones. Tetrahedron Letters, 39 (21), 3617-3620. doi: 10.1016/S0040-4039(98)00564-4 |
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1998 Journal Article Stereoselective synthesis of threo and erythro beta-hydroxy and beta-disubstituted-beta-hydroxy alpha-amino acidsBlaskovich, MA, Evindar, G, Rose, NGW, Wilkinson, S, Luo, Y and Lajoie, GA (1998). Stereoselective synthesis of threo and erythro beta-hydroxy and beta-disubstituted-beta-hydroxy alpha-amino acids. Journal of Organic Chemistry, 63 (11), 3631-3646. doi: 10.1021/jo972294l |
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1998 Journal Article Mild conditions for oxazolidin-5-one formationBlaskovich, MA and Kahn, M (1998). Mild conditions for oxazolidin-5-one formation. Synthesis-Stuttgart (4), 379-380. |
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1998 Journal Article Solid-phase preparation of dienesBlaskovich, MA and Kahn, M (1998). Solid-phase preparation of dienes. Journal of Organic Chemistry, 63 (4), 1119-1125. doi: 10.1021/jo9715884 |
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1993 Journal Article Synthesis of a Chiral Serine Aldehyde Equivalent and its Conversion to Chiral Alpha-Amino-Acid DerivativesBlaskovich, MA and Lajoie, GA (1993). Synthesis of a Chiral Serine Aldehyde Equivalent and its Conversion to Chiral Alpha-Amino-Acid Derivatives. Journal of the American Chemical Society, 115 (12), 5021-5030. doi: 10.1021/ja00065a010 |
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1993 Journal Article Stereoselective Synthesis of Allo-Threonine and Beta-H-2-Allo-Threonine From ThreonineBlaskovich, MA and Lajoie, GA (1993). Stereoselective Synthesis of Allo-Threonine and Beta-H-2-Allo-Threonine From Threonine. Tetrahedron Letters, 34 (24), 3837-3840. doi: 10.1016/S0040-4039(00)79241-0 |
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1991 Journal Article Simple and Convenient Synthesis of Tert-Butyl Ethers of Fmoc-Serine, Fmoc-Threonine, and Fmoc-TyrosineAdamson, JG, Blaskovich, MA, Groenevelt, H and Lajoie, GA (1991). Simple and Convenient Synthesis of Tert-Butyl Ethers of Fmoc-Serine, Fmoc-Threonine, and Fmoc-Tyrosine. Journal of Organic Chemistry, 56 (10), 3447-3449. doi: 10.1021/jo00010a050 |
