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2009

Journal Article

Click peptide by use of the O-acyl isopeptide method: Production of Amyloid Beta peptide from water-soluble analogue

Taniguchi, Atsuhiko, Sohma, Youhei, Skwarczynski, Mariusz, Okada, Takuma, Ikeda, Keisuke, Prakash, Halan, Mukai, Hidehito, Kimura, Tooru, Hayashi, Yoshio, Hirota, Shun, Matsuzaki, Katsumi and Kiso, Yoshiaki (2009). Click peptide by use of the O-acyl isopeptide method: Production of Amyloid Beta peptide from water-soluble analogue. Peptide Science, 397-400.

Click peptide by use of the O-acyl isopeptide method: Production of Amyloid Beta peptide from water-soluble analogue

2008

Journal Article

Controlled production of amyloid beta peptide from a photo-triggered, water-soluble precursor "click peptide"

Taniguchi, Atsuhiko, Skwarczynski, Mariusz, Sohma, Youhei, Okada, Takuma, Ikeda, Keisuke, Prakash, Halan, Mukai, Hidehito, Hayashi, Yoshio, Kimura, Tooru, Hirota, Shun, Matsuzaki, Katsumi and Kiso, Yoshiaki (2008). Controlled production of amyloid beta peptide from a photo-triggered, water-soluble precursor "click peptide". ChemBioChem, 9 (18), 3055-3065. doi: 10.1002/cbic.200800503

Controlled production of amyloid beta peptide from a photo-triggered, water-soluble precursor "click peptide"

2008

Journal Article

Development of novel water-soluble photocleavable protective group and its application for design of photoresponsive paclitaxel prodrugs

Noguchi, Mayo, Skwarczynski, Mariusz, Prakash, Halan, Hirota, Shun, Kimura, Tooru, Hayashi, Yoshio and Kiso, Yoshiaki (2008). Development of novel water-soluble photocleavable protective group and its application for design of photoresponsive paclitaxel prodrugs. Bioorganic and Medicinal Chemistry, 16 (10), 5389-5397. doi: 10.1016/j.bmc.2008.04.022

Development of novel water-soluble photocleavable protective group and its application for design of photoresponsive paclitaxel prodrugs

2007

Journal Article

Application of the O-N intramolecular acyl migration reaction in medicinal chemistry

Skwarczynski, Mariusz and Kiso, Yoshiaki (2007). Application of the O-N intramolecular acyl migration reaction in medicinal chemistry. Current Medicinal Chemistry, 14 (26), 2813-2823. doi: 10.2174/092986707782360123

Application of the O-N intramolecular acyl migration reaction in medicinal chemistry

2007

Journal Article

The synthesis of bioactive peptides based on O-Acyl Isopeptide Method: Application of O-acyl isodipeptide units

Abe, Naoko, Fukao, Fukue, Hayashi, Yoshio, Ito, Nui, Kimura, Tooru, Kiso, Yoshiaki, Nakamura, Setsuko, Skwarczynski, Mariusz, Sohma, Youhei, Taniguchi, Atsuhiko and Yoshiya, Taku (2007). The synthesis of bioactive peptides based on O-Acyl Isopeptide Method: Application of O-acyl isodipeptide units. Peptide Science: Proceedings of the Japanese Peptide Symposium, 44, 187-190.

The synthesis of bioactive peptides based on O-Acyl Isopeptide Method: Application of O-acyl isodipeptide units

2007

Journal Article

"O-acyl isopeptide method" for peptide synthesis: Synthesis of forty kinds of "O-acyl isodipeptide unit" Boc-Ser/Thr(Fmoc-Xaa)-OH

Yoshiya, Taku, Taniguchi, Atsuhiko, Sohma, Youhei, Fukao, Fukue, Nakamura, Setsuko, Abe, Naoko, Ito, Nui, Skwarczynski, Mariusz, Kimura, Tooru, Hayashi, Yoshio and Kiso, Yoshiaki (2007). "O-acyl isopeptide method" for peptide synthesis: Synthesis of forty kinds of "O-acyl isodipeptide unit" Boc-Ser/Thr(Fmoc-Xaa)-OH. Organic and Biomolecular Chemistry, 5 (11), 1720-1730. doi: 10.1039/b702284k

"O-acyl isopeptide method" for peptide synthesis: Synthesis of forty kinds of "O-acyl isodipeptide unit" Boc-Ser/Thr(Fmoc-Xaa)-OH

2007

Conference Publication

Development of new photoresponsive paclitaxel prodrug

Noguchi, Mayo, Skwarczynski, Mariusz, Prakash, Halan, Hirota, Shun, Kimura, Tooru, Hayashi, Yoshio and Kiso, Yoshiaki (2007). Development of new photoresponsive paclitaxel prodrug. 第44回 ペプチド討論会 (44th Japanese Peptide Symposium), Toyama, Toyama Prefecture, Japan, 7-9 November 2007. Osaka, Japan: Protein Research Foundation.

Development of new photoresponsive paclitaxel prodrug

2007

Conference Publication

Synthesis of a Novel Water-Soluble Paclitaxel Prodrug, Arginine-Isotaxel, and its Physicochemical and Caco-2 Transport Properties

Suehisa, Y., Noguchi, M., Skwarczynski, M., Yamamoto, A., Kiso, Y., Hayashi, Y. and Fujita, T. (2007). Synthesis of a Novel Water-Soluble Paclitaxel Prodrug, Arginine-Isotaxel, and its Physicochemical and Caco-2 Transport Properties. 8th Annual Meeting of the International Society for Study of Xenobiotics, Sendai, Japan, 9-12 October 2007. PHILADELPHIA: Informa Healthcare.

Synthesis of a Novel Water-Soluble Paclitaxel Prodrug, Arginine-Isotaxel, and its Physicochemical and Caco-2 Transport Properties

2006

Journal Article

Paclitaxel prodrugs: Toward smarter delivery of anticancer agents

Skwarczynski, Mariusz, Hayashi, Yoshio and Kiso, Yoshiaki (2006). Paclitaxel prodrugs: Toward smarter delivery of anticancer agents. J. Med. Chem., 49 (25), 7253-7269. doi: 10.1021/jm0602155

Paclitaxel prodrugs: Toward smarter delivery of anticancer agents

2006

Journal Article

'Click peptide': A novel 'O-acyl isopeptide method' for peptide synthesis and chemical biology-oriented synthesis of amyloid beta peptide analogues

Sohma, Youhei, Taniguchi, Atsuhiko, Yoshiya, Taku, Chiyomori, Yousuke, Fukao, Fukue, Nakamura, Setsuko, Skwarczynski, Mariusz, Okada, Takuma, Ikeda, Keisuke, Hayashi, Yoshio, Kimura, Tooru, Hirota, Shun, Matsuzaki, Katsumi and Kiso, Yoshiaki (2006). 'Click peptide': A novel 'O-acyl isopeptide method' for peptide synthesis and chemical biology-oriented synthesis of amyloid beta peptide analogues. Journal of Peptide Science, 12 (12), 823-828. doi: 10.1002/psc.817

'Click peptide': A novel 'O-acyl isopeptide method' for peptide synthesis and chemical biology-oriented synthesis of amyloid beta peptide analogues

2006

Journal Article

Application of intramolecular carbonate-carbamate migration

Skwarczynski, M., Noguchi, M., Sohma, Y., Kimura, T., Hayashi, Y. and Kiso, Y. (2006). Application of intramolecular carbonate-carbamate migration. Chimica Oggi, 24 (6), 30-32.

Application of intramolecular carbonate-carbamate migration

2006

Journal Article

Development of first photoresponsive prodrug of paclitaxel

Skwarczynski, Mariusz, Noguchi, Mayo, Hirota. Shun, Sohma, Youhei, Kimura, Tooru, Hayashi, Yoshio and Kiso, Yoshiaki (2006). Development of first photoresponsive prodrug of paclitaxel. Bioorganic and Medicinal Chemistry Letters, 16 (17), 4492-4496. doi: 10.1016/j.bmcl.2006.06.030

Development of first photoresponsive prodrug of paclitaxel

2006

Journal Article

'O-Acyl isopeptide method' for the efficient synthesis of difficult sequence-containing peptides: Use of 'O-acyl isodipeptide unit'

Sohma, Youhei, Taniguchi, Atsuhiko, Skwarczynski, Mariusz, Yoshiya, Taku, Fukao, Fukue, Kimura, Tooru, Hayashi, Yoshio and Kiso, Yoshiaki (2006). 'O-Acyl isopeptide method' for the efficient synthesis of difficult sequence-containing peptides: Use of 'O-acyl isodipeptide unit'. Tetrahedron Letters, 47 (18), 3013-3017. doi: 10.1016/j.tetlet.2006.03.017

'O-Acyl isopeptide method' for the efficient synthesis of difficult sequence-containing peptides: Use of 'O-acyl isodipeptide unit'

2006

Journal Article

O-N intramolecular alkoxycarbonyl migration of typical protective groups in hydroxyamino acids

Skwarczynski, Mariusz, Sohma, Youhei, Noguchi, Mayo, Kimura, Tooru, Hayashi, Yoshio and Kiso, Yoshiaki (2006). O-N intramolecular alkoxycarbonyl migration of typical protective groups in hydroxyamino acids. Journal of Organic Chemistry, 71 (6), 2542-2545. doi: 10.1021/jo0525579

O-N intramolecular alkoxycarbonyl migration of typical protective groups in hydroxyamino acids

2005

Journal Article

No auxiliary, no byproduct strategy for water-soluble prodrugs of taxoids: Scope and limitation of O-N intramolecular acyl and acyloxy migration reactions

Skwarczynski, Mariusz, Sohma, Youhei, Noguchi, Mayo, Kimura, Maiko, Hayashi, Yoshio, Hamada, Yoshio, Kimura, Tooru and Kiso, Yoshiaki (2005). No auxiliary, no byproduct strategy for water-soluble prodrugs of taxoids: Scope and limitation of O-N intramolecular acyl and acyloxy migration reactions. Journal of Medicinal Chemistry, 48 (7), 2655-2666. doi: 10.1021/jm049344g

No auxiliary, no byproduct strategy for water-soluble prodrugs of taxoids: Scope and limitation of O-N intramolecular acyl and acyloxy migration reactions

2004

Conference Publication

O-N intramolecular acyl migration reaction in the development of prodrugs and the synthesis of difficult sequence-containing bioactive peptides

Sohma, Y, Hayashi, Y, Skwarczynski, M, Hamada, Y, Sasaki, M, Kimura, T and Kiso, Y (2004). O-N intramolecular acyl migration reaction in the development of prodrugs and the synthesis of difficult sequence-containing bioactive peptides. 9th Naples Workshop on Bioactive Peptides, Naples Italy, May 08-11, 2004. MALDEN: WILEY-BLACKWELL. doi: 10.1002/bip.20136

O-N intramolecular acyl migration reaction in the development of prodrugs and the synthesis of difficult sequence-containing bioactive peptides

2003

Journal Article

O-N intramolecular acyl migration strategy in water-soluble prodrugs of taxoids

Skwarczynski, M, Sohma, Y, Kimura, M, Hayashi, Y, Kimura, T and Kiso, Y (2003). O-N intramolecular acyl migration strategy in water-soluble prodrugs of taxoids. Bioorganic & Medicinal Chemistry Letters, 13 (24), 4441-4444. doi: 10.1016/j.bmcl.2003.09.020

O-N intramolecular acyl migration strategy in water-soluble prodrugs of taxoids

2003

Journal Article

A novel approach of water-soluble paclitaxel prodrug with no auxiliary and no byproduct: Design and synthesis of isotaxel

Hayashi, Y, Skwarczynski, M, Hamada, Y, Sohma, Y, Kimura, T and Kiso, Y (2003). A novel approach of water-soluble paclitaxel prodrug with no auxiliary and no byproduct: Design and synthesis of isotaxel. Journal of Medicinal Chemistry, 46 (18), 3782-3784. doi: 10.1021/jm034112n

A novel approach of water-soluble paclitaxel prodrug with no auxiliary and no byproduct: Design and synthesis of isotaxel

2003

Journal Article

Mercuric triflate catalyzed hydroxylative carbocyclization of 1,6-enynes

Nishizawa, M, Yadav, VK, Skwarczynski, M, Takao, H, Imagawa, H and Sugihara, T (2003). Mercuric triflate catalyzed hydroxylative carbocyclization of 1,6-enynes. Organic Letters, 5 (10), 1609-1611. doi: 10.1021/ol034201u

Mercuric triflate catalyzed hydroxylative carbocyclization of 1,6-enynes

2002

Journal Article

Mercuric triflate-TMU catalyzed hydration of terminal alkyne to give methyl ketone under mild conditions

Nishizawa, M, Skwarczynski, M, Imagawa, H and Sugihara, T (2002). Mercuric triflate-TMU catalyzed hydration of terminal alkyne to give methyl ketone under mild conditions. Chemistry Letters, 31 (1), 12-13. doi: 10.1246/cl.2002.12

Mercuric triflate-TMU catalyzed hydration of terminal alkyne to give methyl ketone under mild conditions