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2005

Journal Article

No auxiliary, no byproduct strategy for water-soluble prodrugs of taxoids: Scope and limitation of O-N intramolecular acyl and acyloxy migration reactions

Skwarczynski, Mariusz, Sohma, Youhei, Noguchi, Mayo, Kimura, Maiko, Hayashi, Yoshio, Hamada, Yoshio, Kimura, Tooru and Kiso, Yoshiaki (2005). No auxiliary, no byproduct strategy for water-soluble prodrugs of taxoids: Scope and limitation of O-N intramolecular acyl and acyloxy migration reactions. Journal of Medicinal Chemistry, 48 (7), 2655-2666. doi: 10.1021/jm049344g

No auxiliary, no byproduct strategy for water-soluble prodrugs of taxoids: Scope and limitation of O-N intramolecular acyl and acyloxy migration reactions

2004

Conference Publication

O-N intramolecular acyl migration reaction in the development of prodrugs and the synthesis of difficult sequence-containing bioactive peptides

Sohma, Y, Hayashi, Y, Skwarczynski, M, Hamada, Y, Sasaki, M, Kimura, T and Kiso, Y (2004). O-N intramolecular acyl migration reaction in the development of prodrugs and the synthesis of difficult sequence-containing bioactive peptides. 9th Naples Workshop on Bioactive Peptides, Naples Italy, May 08-11, 2004. MALDEN: WILEY-BLACKWELL. doi: 10.1002/bip.20136

O-N intramolecular acyl migration reaction in the development of prodrugs and the synthesis of difficult sequence-containing bioactive peptides

2003

Journal Article

O-N intramolecular acyl migration strategy in water-soluble prodrugs of taxoids

Skwarczynski, M, Sohma, Y, Kimura, M, Hayashi, Y, Kimura, T and Kiso, Y (2003). O-N intramolecular acyl migration strategy in water-soluble prodrugs of taxoids. Bioorganic & Medicinal Chemistry Letters, 13 (24), 4441-4444. doi: 10.1016/j.bmcl.2003.09.020

O-N intramolecular acyl migration strategy in water-soluble prodrugs of taxoids

2003

Journal Article

A novel approach of water-soluble paclitaxel prodrug with no auxiliary and no byproduct: Design and synthesis of isotaxel

Hayashi, Y, Skwarczynski, M, Hamada, Y, Sohma, Y, Kimura, T and Kiso, Y (2003). A novel approach of water-soluble paclitaxel prodrug with no auxiliary and no byproduct: Design and synthesis of isotaxel. Journal of Medicinal Chemistry, 46 (18), 3782-3784. doi: 10.1021/jm034112n

A novel approach of water-soluble paclitaxel prodrug with no auxiliary and no byproduct: Design and synthesis of isotaxel

2003

Journal Article

Mercuric triflate catalyzed hydroxylative carbocyclization of 1,6-enynes

Nishizawa, M, Yadav, VK, Skwarczynski, M, Takao, H, Imagawa, H and Sugihara, T (2003). Mercuric triflate catalyzed hydroxylative carbocyclization of 1,6-enynes. Organic Letters, 5 (10), 1609-1611. doi: 10.1021/ol034201u

Mercuric triflate catalyzed hydroxylative carbocyclization of 1,6-enynes

2002

Journal Article

Mercuric triflate-TMU catalyzed hydration of terminal alkyne to give methyl ketone under mild conditions

Nishizawa, M, Skwarczynski, M, Imagawa, H and Sugihara, T (2002). Mercuric triflate-TMU catalyzed hydration of terminal alkyne to give methyl ketone under mild conditions. Chemistry Letters, 31 (1), 12-13. doi: 10.1246/cl.2002.12

Mercuric triflate-TMU catalyzed hydration of terminal alkyne to give methyl ketone under mild conditions

1999

Journal Article

Enantioselective hydrolysis of 1-butyryloxyalkylphosphonates by lipolytic microorganisms: Pseudomonas fluorescens and Penicillium citrinum

Skwarczynski, M, Lejczak, B and Kafarski, P (1999). Enantioselective hydrolysis of 1-butyryloxyalkylphosphonates by lipolytic microorganisms: Pseudomonas fluorescens and Penicillium citrinum. Chirality, 11 (2), 109-114. doi: 10.1002/(SICI)1520-636X(1999)11:23.0.CO;2-T

Enantioselective hydrolysis of 1-butyryloxyalkylphosphonates by lipolytic microorganisms: Pseudomonas fluorescens and Penicillium citrinum

1996

Journal Article

Accurate assay of enantiopurity of 1-hydroxy- and 2-hydroxyalkylphosphonate esters

Zymanczykduda, E, Skwarczynski, M, Lejczak, B and Kafarski, P (1996). Accurate assay of enantiopurity of 1-hydroxy- and 2-hydroxyalkylphosphonate esters. Tetrahedron-Asymmetry, 7 (5), 1277-1280. doi: 10.1016/0957-4166(96)00143-7

Accurate assay of enantiopurity of 1-hydroxy- and 2-hydroxyalkylphosphonate esters

1996

Journal Article

The Use of Lypolitic Microorganisms Pseudomonas fluorescens and Penicillium citrinum for the Preparation of Optically Active 1 -Hydroxyalkylphosphonates

Lejczak, Barbara, Haliniarz, Ewa, Skwarczynski, Mariusz and Kafarski, Pawel (1996). The Use of Lypolitic Microorganisms Pseudomonas fluorescens and Penicillium citrinum for the Preparation of Optically Active 1 -Hydroxyalkylphosphonates. Phosphorus, Sulfur, and Silicon and the Related Elements, 111 (1), 86-86. doi: 10.1080/10426509608054715

The Use of Lypolitic Microorganisms Pseudomonas fluorescens and Penicillium citrinum for the Preparation of Optically Active 1 -Hydroxyalkylphosphonates

1996

Conference Publication

The use of lypolitic microorganisms Pseudomonas fluorescens and Penicillium citrinum for the preparation of optically active 1-hydroxyalkylphosphonates

Lejczak, B, Haliniarz, E, Skwarczynski, M and Kafarski, P (1996). The use of lypolitic microorganisms Pseudomonas fluorescens and Penicillium citrinum for the preparation of optically active 1-hydroxyalkylphosphonates. 13th International Conference on Phosphorus Chemistry (XIIITH ICPC), Jerusalem Israel, Jul 16-21, 1995. READING: GORDON BREACH SCI PUBL LTD.

The use of lypolitic microorganisms Pseudomonas fluorescens and Penicillium citrinum for the preparation of optically active 1-hydroxyalkylphosphonates

1995

Journal Article

Alkylation of Potassium 1-(n-Benzyloxycarbonylamino)alkylphosphonates and Phosphinates in the Presence of 18-Crown-6

Skwarczynski, M and Kafarski, P (1995). Alkylation of Potassium 1-(n-Benzyloxycarbonylamino)alkylphosphonates and Phosphinates in the Presence of 18-Crown-6. Synthetic Communications, 25 (22), 3565-3571. doi: 10.1080/00397919508015491

Alkylation of Potassium 1-(n-Benzyloxycarbonylamino)alkylphosphonates and Phosphinates in the Presence of 18-Crown-6