1997 Journal Article Conformationally constrained cyclic mimetics of protein and peptide surfaces.Wong, A. K., Reid, R. C., Abbenante, J. and Fairlie, D. P. (1997). Conformationally constrained cyclic mimetics of protein and peptide surfaces.. Abstracts of Papers of The American Chemical Society, 214 (1), 388-ORGN. |
1996 Journal Article Structure-activity relationships for macrocyclic peptidomimetic inhibitors of HIV-1 protease.Abbenante, G., Bergman, D. A., Brinkworth, R. I., March, D. R., Reid, R. C., Hunt, P. A., James, I. W., Dancer, R. J., Garnham, B., Stoermer, M. L. and Fairlie, D. P. (1996). Structure-activity relationships for macrocyclic peptidomimetic inhibitors of HIV-1 protease.. Bioorganic & Medicinal Chemistry Letters, 6 (21), 2531-2536. doi: 10.1016/0960-894X(96)00468-4 |
1996 Journal Article Conformational control by thiazole and oxazoline rings in cyclic octapeptides of marine origin. Novel macrocyclic chair and boat conformationsAbbenante, G., Fairlie, D. P., Gahan, L. R., Hanson, G. R., Pierens, G. K. and van den Brenk, A. L. (1996). Conformational control by thiazole and oxazoline rings in cyclic octapeptides of marine origin. Novel macrocyclic chair and boat conformations. Journal of the American Chemical Society, 118 (43), 10384-10388. doi: 10.1021/ja962260f |
1996 Journal Article A novel bicyclic enzyme inhibitor as a consensus peptidomimetic for the receptor-bound conformations of 12 peptidic inhibitors of HIV-1 proteaseReid, Robert C., March, Darren R., Dooley, Michael J., Bergman, Doug A., Abbenante, Giovanni and Fairlie, David P. (1996). A novel bicyclic enzyme inhibitor as a consensus peptidomimetic for the receptor-bound conformations of 12 peptidic inhibitors of HIV-1 protease. Journal of The American Chemical Society, 118 (36), 8511-8517. doi: 10.1021/ja960433v |
1996 Journal Article Structure of a novel protonated oxadiazine: an unusual heterocycle from the cycloaddition of a ketone with nitrilesKennard, Colin H.L., Byriel, Karl A., Woon, Tai Chin and Fairlie, David P. (1996). Structure of a novel protonated oxadiazine: an unusual heterocycle from the cycloaddition of a ketone with nitriles. Chemical Communications (15), 1731-1732. doi: 10.1039/cc9960001731 |
1996 Journal Article Substrate-based cyclic peptidomimetics of Phe-Ile-Val that inhibit HIV-1 protease using a novel enzyme-binding modeMarch, D. R., Abbenante, G., Bergman, D. A., Brinkworth, R. I., Wickramasinghe, W., Begun, J., Martin, J. L. and Fairlie, D. P. (1996). Substrate-based cyclic peptidomimetics of Phe-Ile-Val that inhibit HIV-1 protease using a novel enzyme-binding mode. Journal of The American Chemical Society, 118 (14), 3375-3379. doi: 10.1021/ja953790z |
1996 Journal Article A novel potassium-binding hydrolysis product of ascidiacyclamide, a cyclic peptide isolated from the ascidian lissoclinum patellavan den Brenk, Anna L., Fairlie, David P., Gahan, Lawrence R., Hanson, Graeme R. and Hambley, Trevor W. (1996). A novel potassium-binding hydrolysis product of ascidiacyclamide, a cyclic peptide isolated from the ascidian lissoclinum patella. Inorganic Chemistry, 35 (5), 1095-1100. doi: 10.1021/ic9504755 |
1996 Journal Article Non-peptide inhibitors of HIV-1 protease. Synthesis and structural evaluation of symmetric and non-symmetric naphthalenesulfonic acid analoguesWong M.F., Huang P.P., Brinkworth R.I., Yashiro M., Mohan P., Fairlie D.P., Baba M. and Verma S. (1996). Non-peptide inhibitors of HIV-1 protease. Synthesis and structural evaluation of symmetric and non-symmetric naphthalenesulfonic acid analogues. European Journal of Medicinal Chemistry, 31 (3), 249-255. doi: 10.1016/0223-5234(96)89141-0 |
1996 Conference Publication Cyclic Peptides as Metal Ion ReceptorsCusack, R. M., Abernante, J., Gahan, L. R., Fairlie, D. P. and Hanson, G. R. (1996). Cyclic Peptides as Metal Ion Receptors. RACI Inorganic Division, IC '96, Townsville, Queensland, Australia, 30 June - 4 July, 1996. |
1996 Conference Publication Effects of conformational constraints in cyclic octapeptides of marine originAbbenante, G., Fairlie, D. P., Sokolenko, N., Gahan, L. R., Cusack, R., Hanson, G. R. and Pierens, G. K. (1996). Effects of conformational constraints in cyclic octapeptides of marine origin. 10th Brisbane Organic Chemistry Symposium, Brisbane, QLD, Australia, 29 November 1996. |
1996 Conference Publication Multifrequency EPR studies of the mono- and bi-nuclear copper(II) complexes formed with the marine cyclic octapeptides patellamide D and ascidiacyclamideHanson, G. R., van den Brenk, A. L., Gahan, L. R., Fairlie, D. P. and Hawkins, C. J. (1996). Multifrequency EPR studies of the mono- and bi-nuclear copper(II) complexes formed with the marine cyclic octapeptides patellamide D and ascidiacyclamide. EPR-95: Electron Paramagnetic Resonance 1995 Satellite Workshop Meeting of the 12th International Society of Magnetic Resonance Conference (ISMAR'95), Sydney, NSW, Australia, 13-15 July 1995. Berlin, Germany: Springer Wien. |
1995 Journal Article Hydroxyquinones are competitive non-peptide inhibitors of HIV-1 proteinaseBrinkworth R.I. and Fairlie D.P. (1995). Hydroxyquinones are competitive non-peptide inhibitors of HIV-1 proteinase. Biochimica et Biophysica Acta (BBA)/Protein Structure and Molecular, 1253 (1), 5-8. doi: 10.1016/0167-4838(95)00183-U |
1995 Journal Article Regioselective Structural and Functional Mimicry of Peptides - Design of Hydrolytically-Stable Cyclic Peptidomimetic Inhibitors of Hiv-1 ProteaseAbbenante, G, March, DR, Bergman, DA, Hunt, PA, Garnham, B, Dancer, RJ, Martin, JL and Fairlie, DP (1995). Regioselective Structural and Functional Mimicry of Peptides - Design of Hydrolytically-Stable Cyclic Peptidomimetic Inhibitors of Hiv-1 Protease. Journal of the American Chemical Society, 117 (41), 10220-10226. doi: 10.1021/ja00146a007 |
1995 Journal Article Nmr Solution Structure of the Rna-Binding Peptide From Human-Immunodeficiency-Virus (type-1) RevScanlon, MJ, Fairlie, DP, Craik, DJ, Englebretsen, DR and West, ML (1995). Nmr Solution Structure of the Rna-Binding Peptide From Human-Immunodeficiency-Virus (type-1) Rev. Biochemistry, 34 (26), 8242-8249. doi: 10.1021/bi00026a005 |
1995 Journal Article A selective and versatile synthesis of substituted chromones via addition of phenols to dimethyl acetylenedicarboxylateStoermer, Martin J. and Fairlie, David P. (1995). A selective and versatile synthesis of substituted chromones via addition of phenols to dimethyl acetylenedicarboxylate. Australian Journal of Chemistry, 48 (3), 677-686. doi: 10.1071/CH9950677 |
1995 Conference Publication The selective binding of tolyporphins to metal ionsAppleton, T. G., Prinsep, M. R., Fairlie, D. P., Lane, I., Hanson, G. R. and Moore, R. E. (1995). The selective binding of tolyporphins to metal ions. 10th National Convention RACI: The Royal Australian Chemical Institute's 10th National Convention: Chemistry Serving Society, Adelaide, SA, Australia, 27 September-2 October 1995. Adelaide, SA, Australia: ICI Australia. |
1995 Journal Article Ammonia and carbon dioxide from urea. A multinuclear NMR study of the activation of urea by platinum(II)Watson A.A. and Fairlie D.P. (1995). Ammonia and carbon dioxide from urea. A multinuclear NMR study of the activation of urea by platinum(II). Inorganic Chemistry, 34 (11), 3087-3092. doi: 10.1021/ic00115a041 |
1995 Conference Publication Multifrequency EPR spectra of Cu(II) and Ag(II) tolyporphinsLane, I., Prinsep, M., Hanson, G. R., Appleton, T. G. and Fairlie, D. (1995). Multifrequency EPR spectra of Cu(II) and Ag(II) tolyporphins. ISMAR 95: Twelfth Conference of the International Society of Magnetic Resonance, Sydney, NSW, Australia, 16-21 July 1995. Philadelphia, PA, U.S.A.: International Society of Magnetic Resonance (ISMAR). |
1995 Journal Article Targeting HIV-1 protease: A test of drug-design methodologiesWest M.L. and Fairlie D.P. (1995). Targeting HIV-1 protease: A test of drug-design methodologies. Trends in Pharmacological Sciences, 16 (2), 67-75. doi: 10.1016/S0165-6147(00)88980-4 |
1995 Journal Article Macrocyclic peptidomimetics - Forcing peptides into bioactive conformationsFairlie D.P., Abenante G. and March D.R. (1995). Macrocyclic peptidomimetics - Forcing peptides into bioactive conformations. Current Medicinal Chemistry, 2 (2), 654-686. doi: 10.2174/0929867302666220218001506 |