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2024

Journal Article

Tobacco, nicotine, and cannabis use and exposure in an Australian Indigenous population during pregnancy: A protocol to measure parental and foetal exposure and outcomes

Ratsch, Angela, Burmeister, Elizabeth A., Bird, Aunty Veronica, Bonner, Aunty Joyce, Miller, Uncle Glen, Speedy, Aunty Marj, Douglas, Graham, Ober, Stevan, Woolcock (nee Geary–Laverty), Ann, Blair (nee Murdoch), Sharly, Weng, Min-Tz, Miles, Jared A. and Steadman, Kathryn J. (2024). Tobacco, nicotine, and cannabis use and exposure in an Australian Indigenous population during pregnancy: A protocol to measure parental and foetal exposure and outcomes. PLoS One, 19 (9) e0300406, 1-22. doi: 10.1371/journal.pone.0300406

Tobacco, nicotine, and cannabis use and exposure in an Australian Indigenous population during pregnancy: A protocol to measure parental and foetal exposure and outcomes

2024

Journal Article

Clinical translation of 3D printed pharmaceuticals

Krueger, Liam, Awad, Atheer, Basit, Abdul W., Goyanes, Alvaro, Miles, Jared A. and Popat, Amirali (2024). Clinical translation of 3D printed pharmaceuticals. Nature Reviews Bioengineering, 2 (10), 1-3. doi: 10.1038/s44222-024-00217-x

Clinical translation of 3D printed pharmaceuticals

2024

Journal Article

The impact of rate of nicotine metabolism, as measured by the nicotine metabolite ratio (NMR), on smoking behaviours during pregnancy: A scoping review

Weng, Min-Tz, Ratsch, Angela, Miles, Jared A., Zheng, Qiuda and Steadman, Kathryn J. (2024). The impact of rate of nicotine metabolism, as measured by the nicotine metabolite ratio (NMR), on smoking behaviours during pregnancy: A scoping review. Health Sciences Review, 12 100186, 1-8. doi: 10.1016/j.hsr.2024.100186

The impact of rate of nicotine metabolism, as measured by the nicotine metabolite ratio (NMR), on smoking behaviours during pregnancy: A scoping review

2023

Journal Article

3D printing tablets for high-precision dose titration of caffeine

Krueger, Liam, Cao, Yuxue, Zheng, Zheng, Ward, Jason, Miles, Jared A. and Popat, Amirali (2023). 3D printing tablets for high-precision dose titration of caffeine. International Journal of Pharmaceutics, 642 123132, 1-9. doi: 10.1016/j.ijpharm.2023.123132

3D printing tablets for high-precision dose titration of caffeine

2023

Journal Article

seco-pregnane glycosides from Australian caustic vine (Cynanchum viminale subsp. australe)

Xue, Yongbo, Savchenko, Andrei I., Agnew-Francis, Kylie A., Miles, Jared A., Holt, Tina, Lu, Hieng, Chow, Sharon, Forster, Paul I., Boyle, Glen M., Ross, Benjamin P., Fischer, Katja, Kutateladze, Andrei G. and Williams, Craig M. (2023). seco-pregnane glycosides from Australian caustic vine (Cynanchum viminale subsp. australe). Journal of Natural Products, 86 (3), 490-497. doi: 10.1021/acs.jnatprod.2c01037

seco-pregnane glycosides from Australian caustic vine (Cynanchum viminale subsp. australe)

2022

Journal Article

3D printing hybrid materials using fused deposition modelling for solid oral dosage forms

Krueger, Liam, Miles, Jared A. and Popat, Amirali (2022). 3D printing hybrid materials using fused deposition modelling for solid oral dosage forms. Journal of Controlled Release, 351, 444-455. doi: 10.1016/j.jconrel.2022.09.032

3D printing hybrid materials using fused deposition modelling for solid oral dosage forms

2022

Journal Article

3D printing: potential clinical applications for personalised solid dose medications

Krueger, Liam, Miles, Jared A., Steadman, Kathryn J., Kumeria, Tushar, Freeman, Christopher R. and Popat, Amirali (2022). 3D printing: potential clinical applications for personalised solid dose medications. Medical Journal of Australia, 216 (2), 64-67. doi: 10.5694/mja2.51381

3D printing: potential clinical applications for personalised solid dose medications

2021

Journal Article

Interaction of opioids with TLR4—mechanisms and ramifications

Gabr, Mai Mahmoud, Saeed, Iqira, Miles, Jared A., Ross, Benjamin P., Shaw, Paul Nicholas, Hollmann, Markus W. and Parat, Marie-Odile (2021). Interaction of opioids with TLR4—mechanisms and ramifications. Cancers, 13 (21) 5274, 5274. doi: 10.3390/cancers13215274

Interaction of opioids with TLR4—mechanisms and ramifications

2021

Journal Article

Discovery of drug-like acetylcholinesterase inhibitors by rapid virtual screening of a 6.9 million compound database

Miles, Jared A., Ng, Jia Hui, Sreenivas, B. Yogi, Courageux, Charlotte, Igert, Alexandre, Dias, José, McGeary, Ross P., Brazzolotto, Xavier and Ross, Benjamin P. (2021). Discovery of drug-like acetylcholinesterase inhibitors by rapid virtual screening of a 6.9 million compound database. Chemical Biology and Drug Design, 97 (5), 1048-1058. doi: 10.1111/cbdd.13825

Discovery of drug-like acetylcholinesterase inhibitors by rapid virtual screening of a 6.9 million compound database

2021

Journal Article

PLGA encapsulated γ-cyclodextrin-meropenem inclusion complex formulation for oral delivery

Raza, Aun, Miles, Jared A., Bruck Sime, Fekade, Ross, Benjamin P., Roberts, Jason A., Popat, Amirali, Kumeria, Tushar and Falconer, James R. (2021). PLGA encapsulated γ-cyclodextrin-meropenem inclusion complex formulation for oral delivery. International Journal of Pharmaceutics, 597 120280, 120280. doi: 10.1016/j.ijpharm.2021.120280

PLGA encapsulated γ-cyclodextrin-meropenem inclusion complex formulation for oral delivery

2021

Journal Article

Protein nanoparticles for enhanced oral delivery of coenzyme-Q10: in vitro and in silico studies

Banun, Vanessa Jane, Rewatkar, Prarthana, Chaudhary, Zanib, Qu, Zhi, Janjua, Taskeen, Patil, Anuja, Wu, Yuao, Ta, Hang T., Bansal, Nidhi, Miles, Jared A., Ross, Benjamin P., Kumeria, Tushar and Popat, Amirali (2021). Protein nanoparticles for enhanced oral delivery of coenzyme-Q10: in vitro and in silico studies. ACS Biomaterials Science and Engineering, 9 (6) acsbiomaterials.0c01354, 2846-2856. doi: 10.1021/acsbiomaterials.0c01354

Protein nanoparticles for enhanced oral delivery of coenzyme-Q10: in vitro and in silico studies

2021

Journal Article

Recent advances in virtual screening for cholinesterase inhibitors

Miles, Jared A. and Ross, Benjamin P. (2021). Recent advances in virtual screening for cholinesterase inhibitors. ACS Chemical Neuroscience, 12 (1) acschemneuro.0c00627, 30-41. doi: 10.1021/acschemneuro.0c00627

Recent advances in virtual screening for cholinesterase inhibitors

2020

Journal Article

Rapid discovery of a selective butyrylcholinesterase inhibitor using structure-based virtual screening

Miles, Jared A., Kapure, Jeevak S., Deora, Girdhar Singh, Courageux, Charlotte, Igert, Alexandre, Dias, José, McGeary, Ross P., Brazzolotto, Xavier and Ross, Benjamin P. (2020). Rapid discovery of a selective butyrylcholinesterase inhibitor using structure-based virtual screening. Bioorganic and Medicinal Chemistry Letters, 30 (24) 127609, 127609. doi: 10.1016/j.bmcl.2020.127609

Rapid discovery of a selective butyrylcholinesterase inhibitor using structure-based virtual screening

2019

Journal Article

Rivastigmine and metabolite analogues with putative Alzheimer’s disease-modifying properties in a Caenorhabditis elegans model

Dighe, Satish N., De la Mora, Eugenio, Chan, Stephen, Kantham, Srinivas, McColl, Gawain, Miles, Jared A., Veliyath, Suresh Kumar, Sreenivas, B. Yogi, Nassar, Zeyad D., Silman, Israel, Sussman, Joel L., Weik, Martin, McGeary, Ross P., Parat, Marie-Odile, Brazzolotto, Xavier and Ross, Benjamin P. (2019). Rivastigmine and metabolite analogues with putative Alzheimer’s disease-modifying properties in a Caenorhabditis elegans model. Communications Chemistry, 2 (1) 35. doi: 10.1038/s42004-019-0133-4

Rivastigmine and metabolite analogues with putative Alzheimer’s disease-modifying properties in a Caenorhabditis elegans model

2017

Journal Article

Effect of the Biphenyl Neolignan Honokiol on Aβ42-Induced Toxicity in Caenorhabditis elegans, Aβ42 Fibrillation, Cholinesterase Activity, DPPH Radicals, and Iron(II) Chelation

Kantham, Srinivas, Chan, Stephen, McColl, Gawain, Miles, Jared A., Veliyath, Suresh Kumar, Deora, Girdhar Singh, Dighe, Satish N., Khabbazi, Samira, Parat, Marie-Odile and Ross, Benjamin P. (2017). Effect of the Biphenyl Neolignan Honokiol on Aβ42-Induced Toxicity in Caenorhabditis elegans, Aβ42 Fibrillation, Cholinesterase Activity, DPPH Radicals, and Iron(II) Chelation. ACS Chemical Neuroscience, 8 (9), 1901-1912. doi: 10.1021/acschemneuro.7b00071

Effect of the Biphenyl Neolignan Honokiol on Aβ42-Induced Toxicity in Caenorhabditis elegans, Aβ42 Fibrillation, Cholinesterase Activity, DPPH Radicals, and Iron(II) Chelation