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2020 Journal Article Rapid discovery of a selective butyrylcholinesterase inhibitor using structure-based virtual screeningMiles, Jared A., Kapure, Jeevak S., Deora, Girdhar Singh, Courageux, Charlotte, Igert, Alexandre, Dias, José, McGeary, Ross P., Brazzolotto, Xavier and Ross, Benjamin P. (2020). Rapid discovery of a selective butyrylcholinesterase inhibitor using structure-based virtual screening. Bioorganic and Medicinal Chemistry Letters, 30 (24) 127609, 127609. doi: 10.1016/j.bmcl.2020.127609 |
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2019 Journal Article Rivastigmine and metabolite analogues with putative Alzheimer’s disease-modifying properties in a Caenorhabditis elegans modelDighe, Satish N., De la Mora, Eugenio, Chan, Stephen, Kantham, Srinivas, McColl, Gawain, Miles, Jared A., Veliyath, Suresh Kumar, Sreenivas, B. Yogi, Nassar, Zeyad D., Silman, Israel, Sussman, Joel L., Weik, Martin, McGeary, Ross P., Parat, Marie-Odile, Brazzolotto, Xavier and Ross, Benjamin P. (2019). Rivastigmine and metabolite analogues with putative Alzheimer’s disease-modifying properties in a Caenorhabditis elegans model. Communications Chemistry, 2 (1) 35. doi: 10.1038/s42004-019-0133-4 |
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2017 Journal Article Effect of the Biphenyl Neolignan Honokiol on Aβ42-Induced Toxicity in Caenorhabditis elegans, Aβ42 Fibrillation, Cholinesterase Activity, DPPH Radicals, and Iron(II) ChelationKantham, Srinivas, Chan, Stephen, McColl, Gawain, Miles, Jared A., Veliyath, Suresh Kumar, Deora, Girdhar Singh, Dighe, Satish N., Khabbazi, Samira, Parat, Marie-Odile and Ross, Benjamin P. (2017). Effect of the Biphenyl Neolignan Honokiol on Aβ42-Induced Toxicity in Caenorhabditis elegans, Aβ42 Fibrillation, Cholinesterase Activity, DPPH Radicals, and Iron(II) Chelation. ACS Chemical Neuroscience, 8 (9), 1901-1912. doi: 10.1021/acschemneuro.7b00071 |