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2014 Conference Publication Mining physicochemical features that contribute to oral bioavailability in peptide middle spacePlisson, Fabien , Lucke, Andrew, Nielsen, Daniel , Stoermer, Martin J. and Fairlie, David (2014). Mining physicochemical features that contribute to oral bioavailability in peptide middle space. European QSAR Symposium, St Petersburg, Russia, September 2014. |
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2013 Journal Article Lithium perchlorate accelerated Friedel-Crafts addition of furans to β-nitrostyrenesStoermer, Martin J., Richter, Hans-Matthias and Kaufmann, Dieter E. (2013). Lithium perchlorate accelerated Friedel-Crafts addition of furans to β-nitrostyrenes. Tetrahedron Letters, 54 (49), 6776-6778. doi: 10.1016/j.tetlet.2013.10.018 |
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2013 Journal Article Downsizing a human inflammatory protein to a small molecule with equal potency and functionalityReid, Robert C., Yau, Mei-Kwan, Singh, Ranee, Hamidon, Johan K., Reed, Anthony N., Chu, Peifei, Suen, Jacky Y., Stoermer, Martin J., Blakeney, Jade S., Lim, Junxian, Faber, Jonathan M. and David P. Fairlie, (2013). Downsizing a human inflammatory protein to a small molecule with equal potency and functionality. Nature Communications, 4 (2802) 2802, 1-9. doi: 10.1038/ncomms3802 |
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2013 Journal Article An interaction between the methyltransferase and RNA dependent RNA polymerase domains of the West Nile virus NS5 proteinTan, Cindy S. E., Hobson-Peters, Jody M., Stoermer, Martin J., Fairlie, David P., Khromykh, Alexander A. and Hall, Roy A. (2013). An interaction between the methyltransferase and RNA dependent RNA polymerase domains of the West Nile virus NS5 protein. Journal of General Virology, 94 (Pt. 9), 1961-1971. doi: 10.1099/vir.0.054395-0 |
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2013 Conference Publication Novel inhibitors of DENV NS2B/NS3pro proteaseChow, Shiao Yun, Stoermer, Martin J., Chappell, Keith J., Young, Paul R. and Fairlie, David P. (2013). Novel inhibitors of DENV NS2B/NS3pro protease. 246th National Meeting of the American-Chemical-Society (ACS), Indianapolis in, Sep 08-12, 2013. WASHINGTON: AMER CHEMICAL SOC. |
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2013 Journal Article Identification and characterization of bi-thiazole-2,2'-diamines as kinase inhibitory scaffoldsNgoei, Kevin R. W., Ng, Dominic C. H., Gooley, Paul R., Fairlie, David P., Stoermer, Martin J. and Bogoyevitch, Marie A. (2013). Identification and characterization of bi-thiazole-2,2'-diamines as kinase inhibitory scaffolds. Biochimica et Biophysica Acta (BBA) - Proteins and Proteomics, 1834 (6), 1077-1088. doi: 10.1016/j.bbapap.2013.02.001 |
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2013 Conference Publication Toward more orally bioavailable inhibitors of phospholipase A(2) GIIA (pla2g2a) to treat chronic inflammationBarbero, Sheila, Reid, Robert C., Stoermer, Martin J., Lohman, Rink J. and Fairlie, David P. (2013). Toward more orally bioavailable inhibitors of phospholipase A(2) GIIA (pla2g2a) to treat chronic inflammation. 246th National Meeting of the American-Chemical-Society (ACS), Indianapolis, IN, United States, 8-12 September 2013. Washington, DC, United States: American Chemical Society. |
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2012 Journal Article Identification of crotonyl glycine in urine of sheep after 48h road transportLi, Juan, Schirra, Horst Joachim, Yu, Yihua, Colgrave, Michelle L., Stoermer, Martin J. and Wijffels, Gene (2012). Identification of crotonyl glycine in urine of sheep after 48h road transport. Journal of Pharmaceutical and Biomedical Analysis, 67–68, 129-136. doi: 10.1016/j.jpba.2012.04.028 |
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2012 Journal Article Structures of peptide agonists for human protease activated receptor 2Stoermer, Martin J., Flanagan, Bernadine, Beyer, Renée L., Madala, Praveen K. and Fairlie, David P. (2012). Structures of peptide agonists for human protease activated receptor 2. Bioorganic and Medicinal Chemistry Letters, 22 (2), 916-919. doi: 10.1016/j.bmcl.2011.12.029 |
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2011 Conference Publication Towards orally bioavailable peptides and peptidomimeticsFairlie, David P., Stoermer, Martin, Lucke, Andrew, Lohman, Rink-Jan, Liu, Ligong and Ruiz-Gomez, Gloria (2011). Towards orally bioavailable peptides and peptidomimetics. 241st National Meeting and Exposition of the American-Chemical-Society (ACS), Anaheim, CA, United States, 27-31 March 2011. Washington, DC, United States: American Chemical Society. |
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2010 Conference Publication Potent inhibitors of West Nile Virus NS2B/NS3 proteaseChappell, K. J., Fairlie, D. P., Gan, C. H., Gupta, P. K., Hu, S., Jensen, C. M., Liebscher, S., Martin, J. L., Robin, G., Stoermer M. J., Xu, W. and Young, P. R. (2010). Potent inhibitors of West Nile Virus NS2B/NS3 protease. 6th General Meeting of the International Proteolysis Society, Gold Coast, QLD, Australia, 26-30 October 2009. Berlin, Germany: Walter De Gruyter. |
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2010 Conference Publication Identification of crotonyl glycine in sheep urine using RP-HPLC, NMR and ESI-MSLi, J., Wijffels, G., Colgrave, M., Stoermer, M.J. and Schirra, H.J. (2010). Identification of crotonyl glycine in sheep urine using RP-HPLC, NMR and ESI-MS. Metabolomics and More - 1st International Metabolomics Symposium in Germany, Freising, Germany, 10-12 March, 2010. |
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2010 Conference Publication Sneaking up on West Nile Virus NS2B/NS3 protease subcellular activity utilising dye-quenched substratesLiebscher, Susan, Chappell, K. J., Stoermer, Martin J., Watterson, Daniel, Webb, Richard I., Khromykh, Alexander A., Fairlie, David P. and Young, Paul R. (2010). Sneaking up on West Nile Virus NS2B/NS3 protease subcellular activity utilising dye-quenched substrates. PlusStrand 2010: The Ninth International Symposium on Positive-Strand RNA Viruses, Atlanta, GA, U.S.A., 17-21 May 2010. |
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2009 Journal Article In silico screening of small molecule libraries using the dengue virus envelope E protein has identified compounds with antiviral activity against multiple flavivirusesKampmann, T., Yennamalli, R., Campbell, P., Stoermer, M. J., Fairlie, D. P., Kobe, B. and Young, P. R. (2009). In silico screening of small molecule libraries using the dengue virus envelope E protein has identified compounds with antiviral activity against multiple flaviviruses. Antiviral Research, 84 (3), 234-241. doi: 10.1016/j.antiviral.2009.09.007 |
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2009 Journal Article Base-sensitivity of arginine alpha-ketoamide inhibitors of serine proteasesStoermer, Martin J., Leung, Donmienne, Young, Paul R. and Fairlie, David P. (2009). Base-sensitivity of arginine alpha-ketoamide inhibitors of serine proteases. Australian Journal of Chemistry, 62 (9), 988-992. doi: 10.1071/CH09150 |
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2009 Journal Article Structure of West Nile virus NS3 protease: Ligand stabilization of the catalytic conformationRobin, Gautier, Chappell, Keith, Stoermer, Martin J., Hu, Shu-Hong, Young, Paul R., Fairlie, David P. and Martin, Jennifer L. (2009). Structure of West Nile virus NS3 protease: Ligand stabilization of the catalytic conformation. Journal of Molecular Biology, 385 (5), 1568-1577. doi: 10.1016/j.jmb.2008.11.026 |
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2009 Conference Publication Potent inhibitors of West Nile Virus NS2B/NS3 proteaseStoermer, Martin , Chappell, Keith J. , Jensen, Christina M. , Liebscher, Susann , Gan, Chun H. , Gupta, Praveer K. , Xu, Wei-Jun , Young, Paul R. , Fairlie, David P. and Watterson, Dan (2009). Potent inhibitors of West Nile Virus NS2B/NS3 protease. 6th General Meeting of the International Proteolysis Society, Gold Coast, QLD, Australia, 26-30 October 2009. |
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2009 Conference Publication Antiviral activity in cell culture of potent inhibitors targeting the West Nile Virus NS2B/NS3 proteaseLiebscher, S., Chappell, K.J., Stoermer, M.J., Fairlie, D.P. and Young, P.R (2009). Antiviral activity in cell culture of potent inhibitors targeting the West Nile Virus NS2B/NS3 protease. 6th General Meeting of the International Proteolysis Society, Gold Coast , QLD, Australia, 26-30 October, 2009. |
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2009 Conference Publication Regulating protein and peptide activated GPCRsFairlie, David P., Madala, Praveen K., Stoermer, Martin J., Suen, Jacky, Barry, Grant and Lohman, Rink-Jan (2009). Regulating protein and peptide activated GPCRs. 229th National Meeting of the American Chemical Society, San Diego, California, 13-17 March 2005. Washington DC, United States: American Chemical Society. |
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2008 Journal Article West Nile Virus NS2B/NS3 protease as an antiviral targetChappell, K. J., Stoermer, M. J., Fairlie, D. P. and Young, P. R. (2008). West Nile Virus NS2B/NS3 protease as an antiviral target. Current Medicinal Chemistry, 15 (27), 2771-2784. doi: 10.2174/092986708786242804 |
