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1996 Journal Article Conformational control by thiazole and oxazoline rings in cyclic octapeptides of marine origin. Novel macrocyclic chair and boat conformationsAbbenante, G., Fairlie, D. P., Gahan, L. R., Hanson, G. R., Pierens, G. K. and van den Brenk, A. L. (1996). Conformational control by thiazole and oxazoline rings in cyclic octapeptides of marine origin. Novel macrocyclic chair and boat conformations. Journal of the American Chemical Society, 118 (43), 10384-10388. doi: 10.1021/ja962260f |
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1996 Journal Article A novel bicyclic enzyme inhibitor as a consensus peptidomimetic for the receptor-bound conformations of 12 peptidic inhibitors of HIV-1 proteaseReid, Robert C., March, Darren R., Dooley, Michael J., Bergman, Doug A., Abbenante, Giovanni and Fairlie, David P. (1996). A novel bicyclic enzyme inhibitor as a consensus peptidomimetic for the receptor-bound conformations of 12 peptidic inhibitors of HIV-1 protease. Journal of The American Chemical Society, 118 (36), 8511-8517. doi: 10.1021/ja960433v |
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1996 Journal Article Structure of a novel protonated oxadiazine: an unusual heterocycle from the cycloaddition of a ketone with nitrilesKennard, Colin H.L., Byriel, Karl A., Woon, Tai Chin and Fairlie, David P. (1996). Structure of a novel protonated oxadiazine: an unusual heterocycle from the cycloaddition of a ketone with nitriles. Chemical Communications (15), 1731-1732. doi: 10.1039/cc9960001731 |
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1996 Journal Article Substrate-based cyclic peptidomimetics of Phe-Ile-Val that inhibit HIV-1 protease using a novel enzyme-binding modeMarch, D. R., Abbenante, G., Bergman, D. A., Brinkworth, R. I., Wickramasinghe, W., Begun, J., Martin, J. L. and Fairlie, D. P. (1996). Substrate-based cyclic peptidomimetics of Phe-Ile-Val that inhibit HIV-1 protease using a novel enzyme-binding mode. Journal of The American Chemical Society, 118 (14), 3375-3379. doi: 10.1021/ja953790z |
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1996 Journal Article A novel potassium-binding hydrolysis product of ascidiacyclamide, a cyclic peptide isolated from the ascidian lissoclinum patellavan den Brenk, Anna L., Fairlie, David P., Gahan, Lawrence R., Hanson, Graeme R. and Hambley, Trevor W. (1996). A novel potassium-binding hydrolysis product of ascidiacyclamide, a cyclic peptide isolated from the ascidian lissoclinum patella. Inorganic Chemistry, 35 (5), 1095-1100. doi: 10.1021/ic9504755 |
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1996 Journal Article Non-peptide inhibitors of HIV-1 protease. Synthesis and structural evaluation of symmetric and non-symmetric naphthalenesulfonic acid analoguesWong M.F., Huang P.P., Brinkworth R.I., Yashiro M., Mohan P., Fairlie D.P., Baba M. and Verma S. (1996). Non-peptide inhibitors of HIV-1 protease. Synthesis and structural evaluation of symmetric and non-symmetric naphthalenesulfonic acid analogues. European Journal of Medicinal Chemistry, 31 (3), 249-255. doi: 10.1016/0223-5234(96)89141-0 |
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1995 Journal Article Hydroxyquinones are competitive non-peptide inhibitors of HIV-1 proteinaseBrinkworth R.I. and Fairlie D.P. (1995). Hydroxyquinones are competitive non-peptide inhibitors of HIV-1 proteinase. Biochimica et Biophysica Acta (BBA)/Protein Structure and Molecular, 1253 (1), 5-8. doi: 10.1016/0167-4838(95)00183-U |
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1995 Journal Article Regioselective Structural and Functional Mimicry of Peptides - Design of Hydrolytically-Stable Cyclic Peptidomimetic Inhibitors of Hiv-1 ProteaseAbbenante, G, March, DR, Bergman, DA, Hunt, PA, Garnham, B, Dancer, RJ, Martin, JL and Fairlie, DP (1995). Regioselective Structural and Functional Mimicry of Peptides - Design of Hydrolytically-Stable Cyclic Peptidomimetic Inhibitors of Hiv-1 Protease. Journal of the American Chemical Society, 117 (41), 10220-10226. doi: 10.1021/ja00146a007 |
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1995 Journal Article Nmr Solution Structure of the Rna-Binding Peptide From Human-Immunodeficiency-Virus (type-1) RevScanlon, MJ, Fairlie, DP, Craik, DJ, Englebretsen, DR and West, ML (1995). Nmr Solution Structure of the Rna-Binding Peptide From Human-Immunodeficiency-Virus (type-1) Rev. Biochemistry, 34 (26), 8242-8249. doi: 10.1021/bi00026a005 |
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1995 Journal Article Macrocyclic peptidomimetics - Forcing peptides into bioactive conformationsFairlie D.P., Abenante G. and March D.R. (1995). Macrocyclic peptidomimetics - Forcing peptides into bioactive conformations. Current Medicinal Chemistry, 2 (2), 654-686. doi: 10.2174/0929867302666220218001506 |
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1995 Journal Article A selective and versatile synthesis of substituted chromones via addition of phenols to dimethyl acetylenedicarboxylateStoermer, Martin J. and Fairlie, David P. (1995). A selective and versatile synthesis of substituted chromones via addition of phenols to dimethyl acetylenedicarboxylate. Australian Journal of Chemistry, 48 (3), 677-686. doi: 10.1071/CH9950677 |
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1995 Journal Article Ammonia and carbon dioxide from urea. A multinuclear NMR study of the activation of urea by platinum(II)Watson A.A. and Fairlie D.P. (1995). Ammonia and carbon dioxide from urea. A multinuclear NMR study of the activation of urea by platinum(II). Inorganic Chemistry, 34 (11), 3087-3092. doi: 10.1021/ic00115a041 |
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1995 Journal Article Targeting HIV-1 protease: A test of drug-design methodologiesWest M.L. and Fairlie D.P. (1995). Targeting HIV-1 protease: A test of drug-design methodologies. Trends in Pharmacological Sciences, 16 (2), 67-75. doi: 10.1016/S0165-6147(00)88980-4 |
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1994 Journal Article Anti-Inflammatory activity of a holothurian (sea cucumber) food supplement in ratsWhitehouse, M. W. and Fairlie, D. P. (1994). Anti-Inflammatory activity of a holothurian (sea cucumber) food supplement in rats. Inflammopharmacology, 2 (4), 411-417. doi: 10.1007/BF02678607 |
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1994 Journal Article Amide-Iminol Tautomerism - Effect of MetalationFairlie, DP, Woo, TC, Wickramasinghe, WA and Willis, AC (1994). Amide-Iminol Tautomerism - Effect of Metalation. Inorganic Chemistry, 33 (26), 6425-6428. doi: 10.1021/ic00104a067 |
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1994 Journal Article Crystal Structure, Electrospray Ionization Mass Spectrometry, Electron Paramagnetic Resonance and Magnetic Susceptibility Study of [Cu2(ascidH2) (1,2-mCO3)(H2O)2].2H2O, the Biscopper (II) Complex of Ascidiacyclamide (ascidH4), a Cyclic Peptide Isolated frvan den Brenk, Anna L., Byriel, Karl A., Fairlie, David P., Gahan, Lawrence R., Hanson, Graeme R., Hawkins, Clifford J., Jones, Alun, Kennard, Colin H. L., Moubaraki, Boujemaa and Murray, Keith S. (1994). Crystal Structure, Electrospray Ionization Mass Spectrometry, Electron Paramagnetic Resonance and Magnetic Susceptibility Study of [Cu2(ascidH2) (1,2-mCO3)(H2O)2].2H2O, the Biscopper (II) Complex of Ascidiacyclamide (ascidH4), a Cyclic Peptide Isolated fr. Inorganic Chemistry, 33 (16), 3549-3557. doi: 10.1021/ic00094a019 |
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1994 Journal Article Binding of copper(II) to the cyclic octapeptide patellamide DVan den Brenk, Anna L., Fairlie, David P., Hanson, Graeme R., Gahan, Lawrence R., Hawkins, Clifford J. and Jones, Alun (1994). Binding of copper(II) to the cyclic octapeptide patellamide D. Inorganic Chemistry, 33 (10), 2280-2289. doi: 10.1021/ic00088a034 |
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1994 Journal Article Anti-inflammatory activity of the isoquinoline alkaloid, tetrandrine, against established adjuvant arthritis in ratsWhitehouse, M. W., Fairlie, D. P. and Thong, Y. H. (1994). Anti-inflammatory activity of the isoquinoline alkaloid, tetrandrine, against established adjuvant arthritis in rats. Agents and Actions, 42 (3-4), 123-127. doi: 10.1007/BF01983477 |
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1993 Journal Article SYNTHESIS, SOLUTION STRUCTURE, AND REACTIVITY OF OXYGEN-BOUND AMIDES ON COBALT(III), (VOL 32, PG 450, 1993)ANGUS, PM, FAIRLIE, DP and JACKSON, WG (1993). SYNTHESIS, SOLUTION STRUCTURE, AND REACTIVITY OF OXYGEN-BOUND AMIDES ON COBALT(III), (VOL 32, PG 450, 1993). Inorganic Chemistry, 32 (19), 4168-4168. doi: 10.1021/ic00071a038 |
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1993 Journal Article Characterisation of TNF-α-related peptides by high-performance liquid chromatography-mass spectrometry and high-performance liquid chromatography-tandem mass spectrometryAlewood P.F., Bailey A.J., Brinkworth R.I., Fairlie D. and Jones A. (1993). Characterisation of TNF-α-related peptides by high-performance liquid chromatography-mass spectrometry and high-performance liquid chromatography-tandem mass spectrometry. Journal of Chromatography A, 646 (1), 185-191. doi: 10.1016/S0021-9673(99)87020-4 |
