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2026 Journal Article Clinical translation of permeation enhancersJanjua, Taskeen Iqbal, Choi, Jeong-Won, Ross, Benjamin P., Gleeson, John P., Mitragotri, Samir and Popat, Amirali (2026). Clinical translation of permeation enhancers. Nature Reviews Materials, 1-21. doi: 10.1038/s41578-026-00954-y |
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2026 Journal Article Piperazine-functionalized nanoparticles enable oral insulin delivery in obese miceCao, Yuxue, Jiang, Xiaofan, Moniruzzaman, Md, Mueller, Alexandra, Janjua, Taskeen Iqbal, Tyagi, Nisha, Qu, Zhi, Wong, Kuan Yau, Feng, Yuran, Ghodasara, Aayushi, Strounina, Ekaterina, Ross, Benjamin P., Kumeria, Tushar, Hasnain, Sumaira Z. and Popat, Amirali (2026). Piperazine-functionalized nanoparticles enable oral insulin delivery in obese mice. Advanced Science, 13 (27) e20918. doi: 10.1002/advs.202520918 |
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2025 Conference Publication Bivalent opioid peptides modulate peripheral mu and delta receptors for pain therapyZhang, Junkai, Robitaille, Melanie, Saifuddin, Danial, Ross, Benjamin P. and Cabot, Peter J. (2025). Bivalent opioid peptides modulate peripheral mu and delta receptors for pain therapy. 2025 ASCEPT and Hypertension Australia Joint Scientific Meeting, Adelaide, SA, Australia, 9-12 December 2025. |
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2025 Conference Publication Targeting peripheral mu and delta opioid receptors with bivalent opioid peptides for pain treatmentZhang, Junkai, Saifuddin, Danial, Robitaille, Melanie, Ross, Benjamin and Cabot, Peter (2025). Targeting peripheral mu and delta opioid receptors with bivalent opioid peptides for pain treatment. Society for Neuroscience (SFN) conference, San Diego, CA, United States, 15-19 November 2025. |
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2025 Journal Article 3D printed tablets for personalised dose titration of prednisone using selective laser sinteringZheng, Zheng, Krueger, Liam, Harrop, Angus C. F., Ross, Benjamin P., Popat, Amirali and Miles, Jared A. (2025). 3D printed tablets for personalised dose titration of prednisone using selective laser sintering. International Journal of Pharmaceutics, 678 125698, 125698. doi: 10.1016/j.ijpharm.2025.125698 |
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2024 Conference Publication Targeting peripheral mu and delta heterodimer receptors with bivalent opioid peptidesZhang, Junkai, Robitaille, Melanie, Saifuddin, Danial, Ross, Benjamin and Cabot, Peter (2024). Targeting peripheral mu and delta heterodimer receptors with bivalent opioid peptides. ASCEPT, APFP & APSA Joint Conference, Melbourne, VIC Australia, 1 - 4 December 2024. |
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2023 Journal Article seco-pregnane glycosides from Australian caustic vine (Cynanchum viminale subsp. australe)Xue, Yongbo, Savchenko, Andrei I., Agnew-Francis, Kylie A., Miles, Jared A., Holt, Tina, Lu, Hieng, Chow, Sharon, Forster, Paul I., Boyle, Glen M., Ross, Benjamin P., Fischer, Katja, Kutateladze, Andrei G. and Williams, Craig M. (2023). seco-pregnane glycosides from Australian caustic vine (Cynanchum viminale subsp. australe). Journal of Natural Products, 86 (3), 490-497. doi: 10.1021/acs.jnatprod.2c01037 |
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2021 Journal Article Interaction of opioids with TLR4—mechanisms and ramificationsGabr, Mai Mahmoud, Saeed, Iqira, Miles, Jared A., Ross, Benjamin P., Shaw, Paul Nicholas, Hollmann, Markus W. and Parat, Marie-Odile (2021). Interaction of opioids with TLR4—mechanisms and ramifications. Cancers, 13 (21) 5274, 5274. doi: 10.3390/cancers13215274 |
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2021 Journal Article Discovery of drug-like acetylcholinesterase inhibitors by rapid virtual screening of a 6.9 million compound databaseMiles, Jared A., Ng, Jia Hui, Sreenivas, B. Yogi, Courageux, Charlotte, Igert, Alexandre, Dias, José, McGeary, Ross P., Brazzolotto, Xavier and Ross, Benjamin P. (2021). Discovery of drug-like acetylcholinesterase inhibitors by rapid virtual screening of a 6.9 million compound database. Chemical Biology and Drug Design, 97 (5), 1048-1058. doi: 10.1111/cbdd.13825 |
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2021 Journal Article pH – responsive colloidal carriers assembled from β-lactoglobulin and epsilon poly-l-lysine for oral drug deliveryPujara, Naisarg, Giri, Rabina, Yau Wong, Kuan, Qu, Zhi, Rewatkar, Prarthana, Moniruzzaman, Md., Begun, Jakob, Ross, Benjamin P., McGuckin, Michael and Popat, Amirali (2021). pH – responsive colloidal carriers assembled from β-lactoglobulin and epsilon poly-l-lysine for oral drug delivery. Journal of Colloid and Interface Science, 589, 45-55. doi: 10.1016/j.jcis.2020.12.054 |
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2021 Journal Article PLGA encapsulated γ-cyclodextrin-meropenem inclusion complex formulation for oral deliveryRaza, Aun, Miles, Jared A., Bruck Sime, Fekade, Ross, Benjamin P., Roberts, Jason A., Popat, Amirali, Kumeria, Tushar and Falconer, James R. (2021). PLGA encapsulated γ-cyclodextrin-meropenem inclusion complex formulation for oral delivery. International Journal of Pharmaceutics, 597 120280, 120280. doi: 10.1016/j.ijpharm.2021.120280 |
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2021 Journal Article Protein nanoparticles for enhanced oral delivery of coenzyme-Q10: in vitro and in silico studiesBanun, Vanessa Jane, Rewatkar, Prarthana, Chaudhary, Zanib, Qu, Zhi, Janjua, Taskeen, Patil, Anuja, Wu, Yuao, Ta, Hang T., Bansal, Nidhi, Miles, Jared A., Ross, Benjamin P., Kumeria, Tushar and Popat, Amirali (2021). Protein nanoparticles for enhanced oral delivery of coenzyme-Q10: in vitro and in silico studies. ACS Biomaterials Science and Engineering, 9 (6) acsbiomaterials.0c01354, 2846-2856. doi: 10.1021/acsbiomaterials.0c01354 |
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2021 Journal Article Recent advances in virtual screening for cholinesterase inhibitorsMiles, Jared A. and Ross, Benjamin P. (2021). Recent advances in virtual screening for cholinesterase inhibitors. ACS Chemical Neuroscience, 12 (1) acschemneuro.0c00627, 30-41. doi: 10.1021/acschemneuro.0c00627 |
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2020 Journal Article Rapid discovery of a selective butyrylcholinesterase inhibitor using structure-based virtual screeningMiles, Jared A., Kapure, Jeevak S., Deora, Girdhar Singh, Courageux, Charlotte, Igert, Alexandre, Dias, José, McGeary, Ross P., Brazzolotto, Xavier and Ross, Benjamin P. (2020). Rapid discovery of a selective butyrylcholinesterase inhibitor using structure-based virtual screening. Bioorganic and Medicinal Chemistry Letters, 30 (24) 127609, 127609. doi: 10.1016/j.bmcl.2020.127609 |
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2020 Journal Article Oral delivery of β-lactoglobulin nanospheres encapsulated resveratrol alleviates inflammation in Winnie mice with spontaneous ulcerative colitisPujara, Naisarg, Wong, Kuan Yau, Qu, Zhi, Wang, Ran, Moniruzzaman, Md., Rewatkar, Prarthana, Kumeria, Tushar, Ross, Benjamin P., McGuckin, Michael and Popat, Amirali (2020). Oral delivery of β-lactoglobulin nanospheres encapsulated resveratrol alleviates inflammation in Winnie mice with spontaneous ulcerative colitis. Molecular Pharmaceutics, 18 (2) acs.molpharmaceut.0c00048, 627-640. doi: 10.1021/acs.molpharmaceut.0c00048 |
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2020 Journal Article A new selective pharmacological enhancer of the Orai1 Ca2+ channel reveals roles for Orai1 in smooth and skeletal muscle functionsAzimi, Iman, Stevenson, Ralph J., Zhang, Xuexin, Meizoso-Huesca, Aldo, Xin, Ping, Johnson, Martin, Flanagan, Jack U., Chalmers, Silke B., Yoast, Ryan E., Kapure, Jeevak S., Ross, Benjamin P., Vetter, Irina, Ashton, Mark R., Launikonis, Bradley S., Denny, William A., Trebak, Mohamed and Monteith, Gregory R. (2020). A new selective pharmacological enhancer of the Orai1 Ca2+ channel reveals roles for Orai1 in smooth and skeletal muscle functions. ACS Pharmacology and Translational Science, 3 (1) acsptsci.9b00081, 135-147. doi: 10.1021/acsptsci.9b00081 |
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2019 Journal Article Rationally designed dendritic silica nanoparticles for oral delivery of exenatideAbeer, Muhammad Mustafa, Meka, Anand Kumar, Pujara, Naisarg, Kumeria, Tushar, Strounina, Ekaterina, Nunes, Rute, Costa, Ana, Sarmento, Bruno, Hasnain, Sumaira Z., Ross, Benjamin P. and Popat, Amirali (2019). Rationally designed dendritic silica nanoparticles for oral delivery of exenatide. Pharmaceutics, 11 (8) 418, 418. doi: 10.3390/pharmaceutics11080418 |
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2019 Journal Article Smad linker region phosphorylation is a signalling pathway in its own right and not only a modulator of canonical TGF-β signallingKamato, Danielle, Do, Bich Hang, Osman, Narin, Ross, Benjamin P., Mohamed, Raafat, Xu, Suowen and Little, Peter J. (2019). Smad linker region phosphorylation is a signalling pathway in its own right and not only a modulator of canonical TGF-β signalling. Cellular and Molecular Life Sciences, 77 (2), 243-251. doi: 10.1007/s00018-019-03266-3 |
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2019 Journal Article A brain-permeable inhibitor of the neurodegenerative disease target kynurenine 3-monooxygenase prevents accumulation of neurotoxic metabolitesZhang, Shaowei, Sakuma, Michiyo, Deora, Girdhar S., Levy, Colin W., Klausing, Alex, Breda, Carlo, Read, Kevin D., Edlin, Chris D., Ross, Benjamin P., Wright Muelas, Marina, Day, Philip J., O’Hagan, Stephen, Kell, Douglas B., Schwarcz, Robert, Leys, David, Heyes, Derren J., Giorgini, Flaviano and Scrutton, Nigel S. (2019). A brain-permeable inhibitor of the neurodegenerative disease target kynurenine 3-monooxygenase prevents accumulation of neurotoxic metabolites. Communications Biology, 2 (1) 271, 271. doi: 10.1038/s42003-019-0520-5 |
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2019 Journal Article Brain delivery of thyrotropin-releasing hormone via a novel prodrug approachProkai-Tatrai, Katalin, De La Cruz, Daniel L., Nguyen, Vien, Ross, Benjamin P., Toth, Istvan and Prokai, Laszlo (2019). Brain delivery of thyrotropin-releasing hormone via a novel prodrug approach. Pharmaceutics, 11 (7) 349, 349. doi: 10.3390/pharmaceutics11070349 |