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2013 Journal Article ChemInform abstract: lipoamino acids as major components of absorption promoters in drug deliveryZiora, Zyta M., Blaskovich, Mark A., Toth, Istvan and Cooper, Matthew A. (2013). ChemInform abstract: lipoamino acids as major components of absorption promoters in drug delivery. ChemInform, 44 (43), no-no. doi: 10.1002/chin.201343267 |
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2013 Journal Article Antibiotics in the clinical pipeline in 2013Butler, Mark S., Blaskovich, Mark A. and Cooper, Matthew A. (2013). Antibiotics in the clinical pipeline in 2013. Journal of Antibiotics, 66 (10), 571-591. doi: 10.1038/ja.2013.86 |
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2013 Journal Article Antibacterial serrulatane diterpenes from the Australian native plant Eremophila microthecaBarnes, Emma C., Kavanagh, Angela M., Ramu, Soumya, Blaskovich, Mark A., Cooper, Matthew A. and Davis, Rohan A. (2013). Antibacterial serrulatane diterpenes from the Australian native plant Eremophila microtheca. Phytochemistry, 93, 162-169. doi: 10.1016/j.phytochem.2013.02.021 |
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2012 Journal Article Resolving biofilm infections: current therapy and drug discovery strategiesRanall, Max V., Butler, Mark S., Blaskovich, Mark A. and Cooper, Matthew A. (2012). Resolving biofilm infections: current therapy and drug discovery strategies. Current Drug Targets, 13 (11), 1375-1385. doi: 10.2174/138945012803530251 |
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2012 Journal Article Lipoamino acids as major components of absorption promoters in drug deliveryZiora, Zyta M., Blaskovich, Mark A., Toth, Istvan and Cooper, Matthew A. (2012). Lipoamino acids as major components of absorption promoters in drug delivery. Current Topics in Medicinal Chemistry, 12 (14), 1562-1580. doi: 10.2174/156802612802652448 |
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2009 Journal Article Drug discovery and protein tyrosine phosphatasesBlaskovich, M. A. T. (2009). Drug discovery and protein tyrosine phosphatases. Current Medicinal Chemistry, 16 (17), 2095-2176. doi: 10.2174/092986709788612693 |
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2008 Journal Article A convenient reduction of α-amino acids to 1,2-amino alcohols with retention of optical purityHwang, Sun-Hee, Blaskovich, Mark A. and Kim, Hwa-Ok (2008). A convenient reduction of α-amino acids to 1,2-amino alcohols with retention of optical purity. Open Organic Chemistry Journal, 2 (1), 107-109. doi: 10.2174/1874095200802010107 |
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2005 Journal Article Design, synthesis, and evaluation of potent and selective benzoyleneurea-based inhibitors of protein geranylgeranyltransferase-1Carrico, D, Blaskovich, MA, Bucher, CJ, Sebti, SM and Hamilton, AD (2005). Design, synthesis, and evaluation of potent and selective benzoyleneurea-based inhibitors of protein geranylgeranyltransferase-1. Bioorganic & Medicinal Chemistry, 13 (3), 677-688. doi: 10.1016/j.bmc.2004.10.053 |
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2004 Journal Article In vitro and in vivo antimalarial activity of peptidomimetic protein farnesyltransferase inhibitors with improved membrane permeabilityCarrico, D, Ohkanda, J, Kendrick, H, Yokoyama, K, Blaskovich, MA, Bucher, CJ, Buckner, FS, Van Voorhis, WC, Chakrabarti, D, Croft, SL, Gelb, MH, Sebti, SM and Hamilton, AD (2004). In vitro and in vivo antimalarial activity of peptidomimetic protein farnesyltransferase inhibitors with improved membrane permeability. Bioorganic & Medicinal Chemistry, 12 (24), 6517-6526. doi: 10.1016/j.bmc.2004.09.020 |
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2004 Journal Article Identification of compounds that enhance the anti-lymphoma activity of rituximab using flow cytometric high-content screeningGasparetto, M, Gentry, T, Sebti, S, O'Bryan, E, Nimmanapalli, R, Blaskovich, MA, Bhalla, K, Rizzieri, D, Haaland, P, Dunne, J and Smith, C (2004). Identification of compounds that enhance the anti-lymphoma activity of rituximab using flow cytometric high-content screening. Journal of Immunological Methods, 292 (1-2), 59-71. doi: 10.1016/j.jim.2004.06.003 |
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2003 Journal Article Design and synthesis of phosphotyrosine mimeticsYan, Zheng, Kahn, Michael, Qabar, Maher, Urban, Jan, Kim, Hwa-Ok and Blaskovich, Mark (2003). Design and synthesis of phosphotyrosine mimetics. Bioorganic & Medicinal Chemistry Letters, 13 (12), 2083-2085. doi: 10.1016/S0960-894X(03)00253-1 |
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2002 Journal Article Recent discovery and development of protein tyrosine phosphatase inhibitorsBlaskovich, Mark A. and Kim, Hwa-Ok (2002). Recent discovery and development of protein tyrosine phosphatase inhibitors. Expert Opinion on Therapeutic Patents, 12 (6), 871-905. doi: 10.1517/13543776.12.6.871 |
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2002 Journal Article Preparation of 1-[N-Benzyloxycarbonyl-(1S)-1-amino-2-oxoethyl]-4-methyl-2,6,7-trioxabicyclo-[2.2.2]octaneRose, Nicholas G.W., Blaskovich, Mark A., Evindar, Ghotas, Wilkinson, Scott, Luo, Yue, Reid, C. and Lajoie, Gilles A. (2002). Preparation of 1-[N-Benzyloxycarbonyl-(1S)-1-amino-2-oxoethyl]-4-methyl-2,6,7-trioxabicyclo-[2.2.2]octane. Organic syntheses, 79, 216-221. doi: 10.1002/0471264180.os079.26 |
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2002 Journal Article Preparation of 1-[N-benzyloxycarbonyl-(1S)-1-amino-2-oxoethyl]-4-methyl-2,6,7-trioxabicyclo[2.2.2] octane: [Carbamic acid, [1-(4-methyl-2,6,7-trioxabicyclo[2.2.2]oct-1-yl)-2-oxoethyl]-, phenylmethyl ester, (S)-]Rose, Nicholas G. W., Blaskovich, Mark A., Evindar, Ghotas, Wilkinson, Scott, Luo, Yue, Fishlock, Dan, Reid, Chris, Lajoie, Gilles A., Gordon, Richard S. and Holmes, Andrew B. (2002). Preparation of 1-[N-benzyloxycarbonyl-(1S)-1-amino-2-oxoethyl]-4-methyl-2,6,7-trioxabicyclo[2.2.2] octane: [Carbamic acid, [1-(4-methyl-2,6,7-trioxabicyclo[2.2.2]oct-1-yl)-2-oxoethyl]-, phenylmethyl ester, (S)-]. Organic Syntheses, 79 doi: 10.15227/orgsyn.079.0216 |
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2001 Journal Article Synthesis of enantiomerically enriched beta,gamma-unsaturated-alpha-amino acidsRose, Ngw, Blaskovich, MA, Wong, A and Lajoie, GA (2001). Synthesis of enantiomerically enriched beta,gamma-unsaturated-alpha-amino acids. Tetrahedron, 57 (8), 1497-1507. doi: 10.1016/S0040-4020(00)01146-7 |
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1999 Journal Article Stereoselective synthesis of beta-substituted alpha,beta-diamino acids from beta-hydroxy amino acidsLuo, Y, Blaskovich, MA and Lajoie, GA (1999). Stereoselective synthesis of beta-substituted alpha,beta-diamino acids from beta-hydroxy amino acids. Journal of Organic Chemistry, 64 (16), 6106-6111. doi: 10.1021/jo9904718 |
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1998 Journal Article Highly efficient and versatile synthesis of libraries of constrained beta-strand mimeticsOgbu, CO, Qabar, MN, Boatman, PD, Urban, J, Meara, JP, Ferguson, MD, Tulinsky, J, Lum, C, Babu, S, Blaskovich, MA, Nakanishi, H, Ruan, FQ, Cao, BL, Minarik, R, Little, T, Nelson, S, Nguyen, M, Gall, A and Kahn, M (1998). Highly efficient and versatile synthesis of libraries of constrained beta-strand mimetics. Bioorganic & Medicinal Chemistry Letters, 8 (17), 2321-2326. doi: 10.1016/S0960-894X(98)00420-X |
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1998 Journal Article Polymer-supported acetylide addition to hexa-2,4-dienalBlaskovich, MA and Kahn, M (1998). Polymer-supported acetylide addition to hexa-2,4-dienal. Synthesis-Stuttgart (7), 965-966. |
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1998 Journal Article Stereoselective synthesis of Threo and Erythro beta-hydroxy and beta-disubstituted-beta-hydroxy alpha-amino acids (vol 63, pg 3635, 1998)Blaskovich, MA, Evindar, G, Rose, NGW, Wilkinson, S, Luo, Y and Lajoie, GA (1998). Stereoselective synthesis of Threo and Erythro beta-hydroxy and beta-disubstituted-beta-hydroxy alpha-amino acids (vol 63, pg 3635, 1998). Journal of Organic Chemistry, 63 (13), 4560-4560. doi: 10.1021/jo9849853 |
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1998 Journal Article Stereoselective synthesis of threo and erythro beta-hydroxy and beta-disubstituted-beta-hydroxy alpha-amino acidsBlaskovich, MA, Evindar, G, Rose, NGW, Wilkinson, S, Luo, Y and Lajoie, GA (1998). Stereoselective synthesis of threo and erythro beta-hydroxy and beta-disubstituted-beta-hydroxy alpha-amino acids. Journal of Organic Chemistry, 63 (11), 3631-3646. doi: 10.1021/jo972294l |
