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2010 Journal Article Tetrapeptides, as small-sized peptidic inhibitors; Synthesis and their inhibitory activity against BACE1Kakizawa, Taeko, Hidaka, Koushi, Hamada, Daisuke, Yamaguchi, Ryoji, Uemura, Tsuyoshi, Kitamura, Hitomi, Tagad, Harichandra D., Hamada, Takashi, Ziora, Zyta, Hamada, Yoshio, Kimura, Tooru and Kiso, Yoshiaki (2010). Tetrapeptides, as small-sized peptidic inhibitors; Synthesis and their inhibitory activity against BACE1. Journal of Peptide Science, 16 (6), 257-262. doi: 10.1002/psc.1238 |
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2010 Journal Article In vitro and in vivo evaluation of positively charged liposaccharide derivatives as oral absorption enhancers for the delivery of anionic drugsBergeon, Julie A., Ziora, Zyta M., Abdelrahim, Adel S., Pernevi, Niklas, Moss, Anne R. and Toth, Istvan (2010). In vitro and in vivo evaluation of positively charged liposaccharide derivatives as oral absorption enhancers for the delivery of anionic drugs. Journal of Pharmaceutical Sciences, 99 (5), 2333-2342. doi: 10.1002/jps.21999 |
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2010 Journal Article Thymine, adenine and lipoamino acid based gene delivery systemsSkwarczynski, Mariusz, Ziora, Zyta M., Coles, Daniel J., Lin, I-Chun and Toth, Istvan (2010). Thymine, adenine and lipoamino acid based gene delivery systems. Chemical Communications, 46 (18), 3140-3142. doi: 10.1039/b924371b |
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2009 Journal Article Design and synthesis of a series of novel, cationic liposaccharide derivatives as potential penetration enhancers for oral drug deliveryAbdelrahim, Adel. S., Ziora, Zyta M., Bergeon, Julie A., Moss, Anne R. and Toth, Istvan (2009). Design and synthesis of a series of novel, cationic liposaccharide derivatives as potential penetration enhancers for oral drug delivery. Tetrahedron, 65 (45), 9436-9442. doi: 10.1016/j.tet.2009.08.072 |
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2009 Journal Article Amidoalkylation of Phosphorus Trichloride with Acetamide and Alkyl OxocycloalkanecarboxylatesZiora, Zyta and Kafarski, Pawel (2009). Amidoalkylation of Phosphorus Trichloride with Acetamide and Alkyl Oxocycloalkanecarboxylates. Phosphorus, Sulfur, and Silicon and the Related Elements, 184 (4), 1047-1053. doi: 10.1080/10426500902737356 |
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2007 Journal Article Potent antimalarial activity of 2-aminopyridinium salts, amidines, and guanidinesCalas, Michele, Outtara, Mahama, Piquet, Giles, Ziora, Zyta, Bordat, Y., Ancelin, Marie L., Escale, Roger and Vial, Henri (2007). Potent antimalarial activity of 2-aminopyridinium salts, amidines, and guanidines. Journal of Medicinal Chemistry, 50 (25), 6307-6315. doi: 10.1021/jm0704752 |
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2007 Journal Article Effect of unsaturated bonds in the sn-2 acyl chain of phosphatidylcholine on the membrane-damaging action of Clostridium perfringens alpha-toxin toward liposomesNagahama, Masahiro, Otsuka, Akiko, Oda, Masataka, Singh, Rajesh K., Ziora, Zyta M., Imagawa, Hiroshi, Nishizawa, Mugio and Sakurai, Jun (2007). Effect of unsaturated bonds in the sn-2 acyl chain of phosphatidylcholine on the membrane-damaging action of Clostridium perfringens alpha-toxin toward liposomes. Biochimica et Biophysica Acta (BBA) - Biomembranes, 1768 (11), 2940-2945. doi: 10.1016/j.bbamem.2007.08.016 |
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2007 Journal Article Design and synthesis of BACE1 inhibitors containing a novel norstatine derivative (2R,3R)-3-amino-2-hydroxy-4(phenylthio)butyric acidZiora, Zyta, Kasai, Soko, Hidaka, Koushi, Nagamine, Ayaka, Kimura, Tooru, Hayashi, Yoshio and Kiso, Yoshiaki (2007). Design and synthesis of BACE1 inhibitors containing a novel norstatine derivative (2R,3R)-3-amino-2-hydroxy-4(phenylthio)butyric acid. Bioorganic and Medicinal Chemistry Letters, 17 (6), 1629-1633. doi: 10.1016/j.bmcl.2006.12.097 |
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2006 Journal Article beta-Secretase inhibitors: Modification at the P-4 position and improvement of inhibitory activity in cultured cellsHamada, Yoshio, Igawa, Naoto, Ikari, Hayato, Ziora, Zyta, Nguyen, Jeffrey-Tri, Yamani, Abdellah, Hidaka, Koushi, Kimura, Tooru, Saito, Kazuki, Hayashi, Yoshio, Ebina, Maiko, Ishiura, Shoichi and Kiso, Yoshiaki (2006). beta-Secretase inhibitors: Modification at the P-4 position and improvement of inhibitory activity in cultured cells. Bioorganic and Medicinal Chemistry Letters, 16 (16), 4354-4359. doi: 10.1016/j.bmcl.2006.05.046 |
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2006 Journal Article Small-sized BACE1 inhibitorsZyta, Ziora, Tooru, KImura and Yoshiaki, Kiso (2006). Small-sized BACE1 inhibitors. Drugs of the Future, 31 (1), 53-63. doi: 10.1358/dof.2006.031.01.957326 |
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2006 Journal Article Phenylthionorstatine as a transition-state mimic in BACE1 inhibitorsZiora Zyta, Kasai Soko, Hidaka Koushi, Nagamine Ayaka, Kimura Tooru, Saito K., Hayashi Yoshio and Kiso Yoshiaki (2006). Phenylthionorstatine as a transition-state mimic in BACE1 inhibitors. Peptide Science, 2006, 237-238. |
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2001 Journal Article Synthesis and spectroscopic characterization of protected N-phosphonomethylglycine dipeptidesZiora, Zyta, Kafarski, Pawel, Holband, Jolanta and Wojcik, Grazyna (2001). Synthesis and spectroscopic characterization of protected N-phosphonomethylglycine dipeptides. Journal of Peptide Science, 7 (9), 466-473. doi: 10.1002/psc.340 |
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2001 Journal Article Conformational polymorphism of diethyl 1-(phthalylglycyloxy)-2-phthalylaminoethenephosphonateHolband, J, Wojcik, G, Ziora, Z and Kafarski, P (2001). Conformational polymorphism of diethyl 1-(phthalylglycyloxy)-2-phthalylaminoethenephosphonate. Journal of Molecular Structure, 595 (1-3), 167-174. doi: 10.1016/S0022-2860(01)00521-X |
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2000 Journal Article H-1 NMR studies of rotational isomerism in phosphonic analogues of aspartic acidJedrzejczyk, D, Ziora, Z and Kafarski, P (2000). H-1 NMR studies of rotational isomerism in phosphonic analogues of aspartic acid. Magnetic Resonance in Chemistry, 38 (5), 370-374. doi: 10.1002/1097-458x(200005)38:53.0.co;2-m |
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2000 Journal Article Reactions of N-phthalylamino acid chlorides with trialkyl phosphitesZiora, Zyta, Maly, Alina, Lejczak, Barbara, Kafarski, Pawel, Holband, Jolanta and Wójcik, Grażyna (2000). Reactions of N-phthalylamino acid chlorides with trialkyl phosphites. Heteroatom Chemistry, 11 (3), 232-239. doi: 10.1002/(sici)1098-1071(2000)11:33.0.co;2-u |
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1999 Journal Article Synthesis of triethyl N-formyl-N-phosphonomethylglycinate and diethyl N-formyl-N- phosphonomethylglycine and studies of their rotational conformers by dynamic NMRZiora, Z, Cierpicki, T, Grembecka, J and Kafarski, P (1999). Synthesis of triethyl N-formyl-N-phosphonomethylglycinate and diethyl N-formyl-N- phosphonomethylglycine and studies of their rotational conformers by dynamic NMR. Journal of Chemical Research (2), 68-69A. doi: 10.1039/a806474a |
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1999 Journal Article Reaction of N-Phtalylamino Acid Chlorides with Trialkyl PhosphitesZiora, Zyta, Maly, Alina, Lejczak, Barbara and Kafarski, Paweł (1999). Reaction of N-Phtalylamino Acid Chlorides with Trialkyl Phosphites. Phosphorus, Sulfur, and Silicon and the Related Elements, 147 (1), 145-145. doi: 10.1080/10426509908053553 |
