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2006

Journal Article

beta-Secretase inhibitors: Modification at the P-4 position and improvement of inhibitory activity in cultured cells

Hamada, Yoshio, Igawa, Naoto, Ikari, Hayato, Ziora, Zyta, Nguyen, Jeffrey-Tri, Yamani, Abdellah, Hidaka, Koushi, Kimura, Tooru, Saito, Kazuki, Hayashi, Yoshio, Ebina, Maiko, Ishiura, Shoichi and Kiso, Yoshiaki (2006). beta-Secretase inhibitors: Modification at the P-4 position and improvement of inhibitory activity in cultured cells. Bioorganic and Medicinal Chemistry Letters, 16 (16), 4354-4359. doi: 10.1016/j.bmcl.2006.05.046

beta-Secretase inhibitors: Modification at the P-4 position and improvement of inhibitory activity in cultured cells

2006

Journal Article

Small-sized BACE1 inhibitors

Zyta, Ziora, Tooru, KImura and Yoshiaki, Kiso (2006). Small-sized BACE1 inhibitors. Drugs of the Future, 31 (1), 53-63. doi: 10.1358/dof.2006.031.01.957326

Small-sized BACE1 inhibitors

2006

Journal Article

Phenylthionorstatine as a transition-state mimic in BACE1 inhibitors

Ziora Zyta, Kasai Soko, Hidaka Koushi, Nagamine Ayaka, Kimura Tooru, Saito K., Hayashi Yoshio and Kiso Yoshiaki (2006). Phenylthionorstatine as a transition-state mimic in BACE1 inhibitors. Peptide Science, 2006, 237-238.

Phenylthionorstatine as a transition-state mimic in BACE1 inhibitors

2006

Conference Publication

Modification of P4 position in beta-Secretase (BACE1) inhibitors containing phenylnorstatine

Ziora, Zyta, Shuto, Daisuke, Kasai, Soko, Liu, Ping, Hidaka, Koushi, Igawa, Nagai, Nagamine, Ayaka, Stochaj, Monika, Hamada, Takashi, Kimura, Tooru, Hayashi, Yoshio and Kiso, Yoshiaki (2006). Modification of P4 position in beta-Secretase (BACE1) inhibitors containing phenylnorstatine. 42nd Japanese Peptide Symposium, Osaka, Japan, 27-29 October 2005. Osaka, Japan: Japanese Peptide Society.

Modification of P4 position in beta-Secretase (BACE1) inhibitors containing phenylnorstatine

2004

Conference Publication

A novel approach for the hydrophobic peptides synthesis and purification through O-N intramolecular acyl migration reaction

Sohma, Youhei, Sasaki, Masato, Ziora, Zyta, Takahashi, N., Kimura, Tooru, Hayashi, Yoshio and Kiso, Yoshiaki (2004). A novel approach for the hydrophobic peptides synthesis and purification through O-N intramolecular acyl migration reaction. 18th American Peptide Symposium, Boston, MA, U.S.A., 19-23 July 2003. San Diego, CA, U.S.A.: American Peptide Society.

A novel approach for the hydrophobic peptides synthesis and purification through O-N intramolecular acyl migration reaction

2001

Journal Article

Synthesis and spectroscopic characterization of protected N-phosphonomethylglycine dipeptides

Ziora, Zyta, Kafarski, Pawel, Holband, Jolanta and Wojcik, Grazyna (2001). Synthesis and spectroscopic characterization of protected N-phosphonomethylglycine dipeptides. Journal of Peptide Science, 7 (9), 466-473. doi: 10.1002/psc.340

Synthesis and spectroscopic characterization of protected N-phosphonomethylglycine dipeptides

2001

Journal Article

Conformational polymorphism of diethyl 1-(phthalylglycyloxy)-2-phthalylaminoethenephosphonate

Holband, J, Wojcik, G, Ziora, Z and Kafarski, P (2001). Conformational polymorphism of diethyl 1-(phthalylglycyloxy)-2-phthalylaminoethenephosphonate. Journal of Molecular Structure, 595 (1-3), 167-174. doi: 10.1016/S0022-2860(01)00521-X

Conformational polymorphism of diethyl 1-(phthalylglycyloxy)-2-phthalylaminoethenephosphonate

2000

Journal Article

H-1 NMR studies of rotational isomerism in phosphonic analogues of aspartic acid

Jedrzejczyk, D, Ziora, Z and Kafarski, P (2000). H-1 NMR studies of rotational isomerism in phosphonic analogues of aspartic acid. Magnetic Resonance in Chemistry, 38 (5), 370-374. doi: 10.1002/1097-458x(200005)38:53.0.co;2-m

H-1 NMR studies of rotational isomerism in phosphonic analogues of aspartic acid

2000

Journal Article

Reactions of N-phthalylamino acid chlorides with trialkyl phosphites

Ziora, Zyta, Maly, Alina, Lejczak, Barbara, Kafarski, Pawel, Holband, Jolanta and Wójcik, Grażyna (2000). Reactions of N-phthalylamino acid chlorides with trialkyl phosphites. Heteroatom Chemistry, 11 (3), 232-239. doi: 10.1002/(sici)1098-1071(2000)11:33.0.co;2-u

Reactions of N-phthalylamino acid chlorides with trialkyl phosphites

1999

Journal Article

Synthesis of triethyl N-formyl-N-phosphonomethylglycinate and diethyl N-formyl-N- phosphonomethylglycine and studies of their rotational conformers by dynamic NMR

Ziora, Z, Cierpicki, T, Grembecka, J and Kafarski, P (1999). Synthesis of triethyl N-formyl-N-phosphonomethylglycinate and diethyl N-formyl-N- phosphonomethylglycine and studies of their rotational conformers by dynamic NMR. Journal of Chemical Research (2), 68-69A. doi: 10.1039/a806474a

Synthesis of triethyl N-formyl-N-phosphonomethylglycinate and diethyl N-formyl-N- phosphonomethylglycine and studies of their rotational conformers by dynamic NMR

1999

Journal Article

Reaction of N-Phtalylamino Acid Chlorides with Trialkyl Phosphites

Ziora, Zyta, Maly, Alina, Lejczak, Barbara and Kafarski, Paweł (1999). Reaction of N-Phtalylamino Acid Chlorides with Trialkyl Phosphites. Phosphorus, Sulfur, and Silicon and the Related Elements, 147 (1), 145-145. doi: 10.1080/10426509908053553

Reaction of N-Phtalylamino Acid Chlorides with Trialkyl Phosphites